Page last updated: 2024-09-03

way 100135 and citalopram

way 100135 has been researched along with citalopram in 6 studies

Compound Research Comparison

Studies
(way 100135)
Trials
(way 100135)
Recent Studies (post-2010)
(way 100135)
Studies
(citalopram)
Trials
(citalopram)
Recent Studies (post-2010) (citalopram)
1430345,3481,4242,350

Protein Interaction Comparison

ProteinTaxonomyway 100135 (IC50)citalopram (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.297
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)2.196
AromataseRattus norvegicus (Norway rat)0.0018
Sodium-dependent noradrenaline transporter Homo sapiens (human)2.196
Alpha-1D adrenergic receptorHomo sapiens (human)3.289
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.297
Sodium-dependent serotonin transporterHomo sapiens (human)0.0227
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.0027
Histamine H1 receptorHomo sapiens (human)3.194
5-hydroxytryptamine receptor 2BHomo sapiens (human)1.839
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.1869
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.398
TransporterRattus norvegicus (Norway rat)8.8

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (50.00)18.2507
2000's2 (33.33)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Arborelius, L; Grillner, P; Hacksell, U; Hertel, P; Höök, BB; Nomikos, GG; Svensson, TH1
Auerbach, SB; Hjorth, S1
Hashimoto, S; Inoue, T; Koyama, T1
Höglund, AU; Kommalage, M1
Eckler, JR; Rabin, RA; Rice, KC; Winter, JC1
Csatlósová, K; Dremencov, E; Durišová, B; Ježová, D; Lacinová, L; Moravcíková, L1

Other Studies

6 other study(ies) available for way 100135 and citalopram

ArticleYear
5-HT1A receptor antagonists increase the activity of serotonergic cells in the dorsal raphe nucleus in rats treated acutely or chronically with citalopram.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Citalopram; Electrophysiology; Extracellular Space; Male; Neurons; Piperazines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Synaptic Transmission

1995
Further evidence for the importance of 5-HT1A autoreceptors in the action of selective serotonin reuptake inhibitors.
    European journal of pharmacology, 1994, Aug-01, Volume: 260, Issue:2-3

    Topics: Analysis of Variance; Animals; Antidepressive Agents; Autoreceptors; Citalopram; Hippocampus; Male; Microdialysis; Paroxetine; Pindolol; Piperazines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Stereoisomerism

1994
Effects of the co-administration of 5-HT1A receptor antagonists with an SSRI in conditioned fear stress-induced freezing behavior.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 58, Issue:2

    Topics: Animals; Behavior, Animal; Citalopram; Conditioning, Psychological; Drug Synergism; Fear; Male; Piperazines; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Stress, Physiological

1997
Involvement of spinal serotonin receptors in the regulation of intraspinal acetylcholine release.
    European journal of pharmacology, 2005, Feb-21, Volume: 509, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Amphetamines; Animals; Biguanides; Citalopram; Dose-Response Relationship, Drug; Ketanserin; Male; Microdialysis; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Time Factors

2005
Serotonergic/glutamatergic interactions: potentiation of phencyclidine-induced stimulus control by citalopram.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:3

    Topics: Aminopyridines; Analysis of Variance; Animals; Citalopram; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Indoles; Male; Phencyclidine; Piperazines; Rats; Rats, Inbred F344; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2005
Effect of Physical Exercise and Acute Escitalopram on the Excitability of Brain Monoamine Neurons: In Vivo Electrophysiological Study in Rats.
    The international journal of neuropsychopharmacology, 2017, 07-01, Volume: 20, Issue:7

    Topics: Action Potentials; Analysis of Variance; Animals; Biogenic Monoamines; Brain; Citalopram; Locomotion; Male; Neurons; Physical Conditioning, Animal; Piperazines; Random Allocation; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Time Factors

2017