Page last updated: 2024-10-24

bradykinin receptor activity

Definition

Target type: molecularfunction

Combining with bradykinin to initiate a change in cell activity. [GOC:ai]

Proteins (2)

ProteinDefinitionTaxonomy
B1 bradykinin receptorA B1 bradykinin receptor that is encoded in the genome of human. [PRO:WCB, UniProtKB:P46663]Homo sapiens (human)
B2 bradykinin receptorA B2 bradykinin receptor that is encoded in the genome of human. [PRO:WCB, UniProtKB:P30411]Homo sapiens (human)

Compounds (21)

CompoundDefinitionClassesRoles
amiodaroneamiodarone : A member of the class of 1-benzofurans that is 1-benzofuran substituted by a butyl group at position 2 and a 4-[2-(diethylamino)ethoxy]-3,5-diiodobenzoyl group at position 3. It is a cardiovascular drug used for the treatment of cardiac dysrhythmias.

Amiodarone: An antianginal and class III antiarrhythmic drug. It increases the duration of ventricular and atrial muscle action by inhibiting POTASSIUM CHANNELS and VOLTAGE-GATED SODIUM CHANNELS. There is a resulting decrease in heart rate and in vascular resistance.
1-benzofurans;
aromatic ketone;
organoiodine compound;
tertiary amino compound
cardiovascular drug
diacetylfluorescein
coumarin 153coumarin 153: structure in first source7-aminocoumarinsfluorochrome
2-butyl-6-(butylamino)-1h-benzo(de)isoquinoline-1,3(2h)-dione
coumarin 7coumarin 7: structure in first source
arg-3-hyp-7-phe-bradykininNPC 567: bradykinin receptor antagonist

NPC-567 : A ten-membered oligopeptide comprising D-arginyl, L-arginyl, L-prolyl, (4R)-4-hydroxy-L-prolyl, glycyl, L-phenylalanyl, L-seryl, D-phenylalanyl, L-phenylalanyl and L-arginine residues joined in sequence.
oligopeptidebradykinin receptor antagonist
kallidin, des-arg(10)-kallidin, des-Arg(10)-: includes both L and D isomers of Phe(8)
bradykinin, leu(8)-des-arg(9)-bradykinin, Leu(8)-des-Arg(9)-: RN given refers to (L)-isomer
bradykininoligopeptidehuman blood serum metabolite;
vasodilator agent
tamoxifenstilbenoid;
tertiary amino compound
angiogenesis inhibitor;
antineoplastic agent;
bone density conservation agent;
EC 1.2.3.1 (aldehyde oxidase) inhibitor;
EC 2.7.11.13 (protein kinase C) inhibitor;
estrogen antagonist;
estrogen receptor antagonist;
estrogen receptor modulator
3,7-dichloro-N-[3-(1-imidazolyl)propyl]-6-methoxy-1-benzothiophene-2-carboxamide1-benzothiophenes
fr 173657FR 173657: structure given in first source
fr 190997FR 190997: structure given in first source
bradyzidebradyzide: structure in first source
icatibantoligopeptidebeta-adrenergic antagonist;
bradykinin receptor antagonist;
peptidomimetic
rmp 7RMP 7: a synthetic bradykinin analog; selectively increases uptake of molecular tracers in RG2 glial tumors
cp 195543CP 195543: a potent & selective leukotriene B4 antagonist; structure in first source
cp 105696CP 105696: a leukotriene B4 receptor antagonist; structure in first source
lissamine rhodamine blissamine rhodamine : An organic sodium salt having 4-[3,6-bis(diethylamino)xanthenium-9-yl]benzene-1,3-disulfonate as the counterion.organic sodium saltfluorescent probe;
fluorochrome;
histological dye
eln441958ELN441958: bradykinin B1 Receptor antagonist; structure in first source
nitd 609NITD 609: an antimalarial and coccidiostat; structure in first source