Page last updated: 2024-09-02

zacopride and cocaine

zacopride has been researched along with cocaine in 4 studies

Compound Research Comparison

Studies
(zacopride)
Trials
(zacopride)
Recent Studies (post-2010)
(zacopride)
Studies
(cocaine)
Trials
(cocaine)
Recent Studies (post-2010) (cocaine)
18041632,4611,0969,400

Protein Interaction Comparison

ProteinTaxonomyzacopride (IC50)cocaine (IC50)
Amyloid-beta precursor proteinHomo sapiens (human)0.338
Fatty acid-binding protein, heartHomo sapiens (human)0.367
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0855
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0855
DRattus norvegicus (Norway rat)5.7544
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)5.7544
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.2861
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.4321
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0855
Sodium-dependent serotonin transporterHomo sapiens (human)0.5442
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.8885
Sodium-dependent dopamine transporter Homo sapiens (human)0.3796
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.541
Sodium-dependent dopamine transporterMus musculus (house mouse)0.2
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.05
TransporterRattus norvegicus (Norway rat)3.2277

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hitzemann, R; Svingos, AL1
Barnes, NM; Costall, B; Kelly, ME; Naylor, RJ; Onaivi, ES1
Reith, ME1
Hitzemann, R; McNeish, CS; Strecker, RE; Svingos, AL1

Other Studies

4 other study(ies) available for zacopride and cocaine

ArticleYear
5-HT3 receptor antagonists block cocaine-induced locomotion via a PCPA-sensitive mechanism.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:3

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Dose-Response Relationship, Drug; Fenclonine; Indoles; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Tropanes; Tropisetron

1992
Ketotifen and its analogues reduce aversive responding in the rodent.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:4

    Topics: Animals; Avoidance Learning; Behavior, Animal; Benzamides; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Diazepam; Ethanol; Exploratory Behavior; Granisetron; Indazoles; Ketotifen; Male; Mice; Mice, Inbred Strains; Nicotine; Radioligand Assay; Rats; Rats, Inbred Strains; Serotonin Antagonists; Social Behavior

1990
5-HT3 receptor antagonists attenuate cocaine-induced locomotion in mice.
    European journal of pharmacology, 1990, Sep-21, Volume: 186, Issue:2-3

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Caffeine; Cocaine; Drug Interactions; Indoles; Male; Methysergide; Mice; Mice, Inbred C57BL; Motor Activity; Receptors, Serotonin; Serotonin Antagonists; Tropisetron

1990
The 5-HT3 antagonist zacopride attenuates cocaine-induced increases in extracellular dopamine in rat nucleus accumbens.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chromatography, High Pressure Liquid; Cocaine; Dialysis; Dopamine; Extracellular Space; Homovanillic Acid; Male; Motor Activity; Nucleus Accumbens; Prosencephalon; Rats; Rats, Sprague-Dawley; Serotonin Antagonists

1993