Page last updated: 2024-09-05

tau 284 and ketotifen

tau 284 has been researched along with ketotifen in 3 studies

Compound Research Comparison

Studies
(tau 284)
Trials
(tau 284)
Recent Studies (post-2010)
(tau 284)
Studies
(ketotifen)
Trials
(ketotifen)
Recent Studies (post-2010) (ketotifen)
5218211,212275151

Protein Interaction Comparison

ProteinTaxonomytau 284 (IC50)ketotifen (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.16
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.838
Muscarinic acetylcholine receptor M4Homo sapiens (human)1.009
Muscarinic acetylcholine receptor M5Homo sapiens (human)0.374
Alpha-2A adrenergic receptorHomo sapiens (human)2.187
Muscarinic acetylcholine receptor M1Homo sapiens (human)1.112
Alpha-2B adrenergic receptorHomo sapiens (human)0.71
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)2.537
Muscarinic acetylcholine receptor M3Homo sapiens (human)2.209
D(1A) dopamine receptorHomo sapiens (human)0.872
Histamine H2 receptorHomo sapiens (human)4.129
Alpha-1D adrenergic receptorHomo sapiens (human)3.727
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.031
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.16
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)2.537
Histamine H1 receptorHomo sapiens (human)0.0011
D(3) dopamine receptorHomo sapiens (human)1.963
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.046
5-hydroxytryptamine receptor 6Homo sapiens (human)1.141

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's0 (0.00)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ikezawa, K; Kaminuma, O; Kikkawa, H; Kikuchi, M; Naito, K; Ogawa, K1
Inagaki, N; Koda, A; Nagai, H; Ueno, M1
Kanamitsu, K; Kusuhara, H; Nagaya, Y; Nozaki, Y; Sugiyama, Y1

Other Studies

3 other study(ies) available for tau 284 and ketotifen

ArticleYear
A novel anti-allergic drug, betotastine besilate, suppresses interleukin-5 production by human peripheral blood mononuclear cells.
    Biological & pharmaceutical bulletin, 1998, Volume: 21, Issue:4

    Topics: Adult; Anti-Allergic Agents; Cell Division; Cells, Cultured; Humans; Indicators and Reagents; Interleukin-5; Ketotifen; Male; Middle Aged; Monocytes; Piperidines; Pyridines

1998
Antiallergic action of betotastine besilate (TAU-284) in animal models: A comparison with ketotifen.
    Pharmacology, 1998, Volume: 57, Issue:4

    Topics: Animals; Anti-Allergic Agents; Asthma; Bronchoconstriction; Disease Models, Animal; Eosinophilia; Eosinophils; Female; Guinea Pigs; Histamine H1 Antagonists; Hypersensitivity; Ketotifen; Male; Passive Cutaneous Anaphylaxis; Piperidines; Platelet Activating Factor; Pyridines; Rats; Rats, Wistar

1998
Quantitative prediction of histamine H1 receptor occupancy by the sedative and non-sedative antagonists in the human central nervous system based on systemic exposure and preclinical data.
    Drug metabolism and pharmacokinetics, 2017, Volume: 32, Issue:2

    Topics: Animals; Brain; Central Nervous System; Diphenhydramine; Histamine H1 Antagonists; Humans; Ketotifen; Macaca fascicularis; Male; Mice; Mice, Inbred Strains; Olopatadine Hydrochloride; Piperidines; Positron-Emission Tomography; Pyridines; Receptors, Histamine H1; Time Factors

2017