Page last updated: 2024-09-03

tak 044 and prazosin

tak 044 has been researched along with prazosin in 1 studies

Compound Research Comparison

Studies
(tak 044)
Trials
(tak 044)
Recent Studies (post-2010)
(tak 044)
Studies
(prazosin)
Trials
(prazosin)
Recent Studies (post-2010) (prazosin)
105827,914713682

Protein Interaction Comparison

ProteinTaxonomytak 044 (IC50)prazosin (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)5.87
Interstitial collagenaseHomo sapiens (human)4.036
Alpha-2A adrenergic receptorHomo sapiens (human)2.638
Matrix metalloproteinase-9Homo sapiens (human)6.963
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0008
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)0.0078
Alpha-2B adrenergic receptorHomo sapiens (human)0.29
Alpha-2C adrenergic receptorHomo sapiens (human)0.647
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.0008
Alpha-1D adrenergic receptorHomo sapiens (human)0.0007
Bromodomain-containing protein 2Homo sapiens (human)0.0009
Alpha-1A adrenergic receptorHomo sapiens (human)0.0006
Alpha-1B adrenergic receptorHomo sapiens (human)0.0006
5-hydroxytryptamine receptor 2BHomo sapiens (human)4.118
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0008
5-hydroxytryptamine receptor 7Cavia porcellus (domestic guinea pig)9.9
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.5849
Multidrug and toxin extrusion protein 1Homo sapiens (human)1.6

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Endoh, M; Yang, HT; Zhu, Y1

Other Studies

1 other study(ies) available for tak 044 and prazosin

ArticleYear
Negative chronotropic and inotropic effects of endothelin isopeptides in mammalian cardiac muscle.
    The American journal of physiology, 1997, Volume: 273, Issue:1 Pt 2

    Topics: Animals; Cyclic AMP; Dogs; Endothelin Receptor Antagonists; Endothelin-1; Endothelin-3; Heart Atria; Heart Rate; Heart Ventricles; In Vitro Techniques; Isoproterenol; Male; Mammals; Myocardial Contraction; Myocardium; Peptides, Cyclic; Pertussis Toxin; Prazosin; Rabbits; Receptor, Endothelin A; Receptor, Endothelin B; Virulence Factors, Bordetella

1997
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