Page last updated: 2024-09-02

st 587 and guanabenz

st 587 has been researched along with guanabenz in 2 studies

Compound Research Comparison

Studies
(st 587)
Trials
(st 587)
Recent Studies (post-2010)
(st 587)
Studies
(guanabenz)
Trials
(guanabenz)
Recent Studies (post-2010) (guanabenz)
67004464296

Protein Interaction Comparison

ProteinTaxonomyst 587 (IC50)guanabenz (IC50)
trace amine-associated receptor 1Homo sapiens (human)1.173
Solute carrier family 22 member 1 Homo sapiens (human)4.85
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.204
Alpha-2A adrenergic receptorHomo sapiens (human)0.041
Alpha-2B adrenergic receptorHomo sapiens (human)0.149
Alpha-2C adrenergic receptorHomo sapiens (human)1.106
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)2.068
Amine oxidase [flavin-containing] AHomo sapiens (human)1.787
Alpha-1D adrenergic receptorHomo sapiens (human)0.472
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.392
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.204
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)2.068
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.097

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Kubo, T; Misu, Y; Nagura, J1

Other Studies

2 other study(ies) available for st 587 and guanabenz

ArticleYear
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction

1984
Pharmacological characterization of spinal alpha adrenoceptors related to blood pressure control in rats.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Brain Stem; Clonidine; Dopamine; Guanabenz; Hydroxydopamines; Injections, Spinal; Male; Norepinephrine; Oxidopamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Spinal Cord; Yohimbine

1987