Proteins > trace amine-associated receptor 1
Page last updated: 2024-08-07 22:58:24

trace amine-associated receptor 1

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (25)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
tyramineHomo sapiens (human)IC500.881810
tolazoline hydrochlorideHomo sapiens (human)IC504.742010
hydroxyamphetamine hydrobromideHomo sapiens (human)IC508.844510
tetrahydrozoline hydrochlorideHomo sapiens (human)IC500.157110
naphazoline hydrochlorideHomo sapiens (human)IC501.154010
lysergolHomo sapiens (human)IC504.577010
antazoline hydrochlorideHomo sapiens (human)IC5029.903010
proroxan hydrochlorideHomo sapiens (human)IC501.157520
fenoldopam mesylateHomo sapiens (human)IC508.044010
formetamideHomo sapiens (human)IC502.268010
antazoline phosphateHomo sapiens (human)IC5029.909010
sercHomo sapiens (human)IC506.018010
8-anilino-1,3-dimethyl-7H-purine-2,6-dioneHomo sapiens (human)IC509.394010
N-[3-(2-phenylethyl)-2,4-dihydro-1H-1,3,5-triazin-6-yl]-1,3-benzoxazol-2-amineHomo sapiens (human)IC5014.721010
N-(2-fluorophenyl)-4-phenylmethoxybenzamideHomo sapiens (human)IC5027.705010
4-[5-(2-phenylethyl)-2-sulfanylidene-1,3,5-triazinan-1-yl]benzoic acid ethyl esterHomo sapiens (human)IC500.775510
N-(2-phenylethyl)-5-thiophen-2-yl-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamideHomo sapiens (human)IC501.910010
N1-phenethylhydrazine-1-carbothioamideHomo sapiens (human)IC5010.382010
phenacylamine monohydrochlorideHomo sapiens (human)IC507.415010
(1R,2S)-tranylcypromine hydrochlorideHomo sapiens (human)IC502.097010
2,6-difluoro-N-[2-[3-[(2-fluorophenyl)methylthio]-1-indolyl]ethyl]benzamideHomo sapiens (human)IC5010.289520
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[5-methyl-2-(4-methylphenyl)-4-oxazolyl]methylsulfonyl]ethanoneHomo sapiens (human)IC505.402010
guanabenzHomo sapiens (human)IC501.173010
3-methoxytyramine hydrochlorideHomo sapiens (human)IC5021.614010
1-hydroxy-5-nitro-N-(2-phenylethyl)-4-spiro[benzimidazole-2,1'-cyclohexane]imineHomo sapiens (human)IC508.858010

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
tyramineHomo sapiens (human)EC500.177710
tolazoline hydrochlorideHomo sapiens (human)EC501.011010
hydroxyamphetamine hydrobromideHomo sapiens (human)EC501.445010
tetrahydrozoline hydrochlorideHomo sapiens (human)EC500.154410
naphazoline hydrochlorideHomo sapiens (human)EC500.140210
lysergolHomo sapiens (human)EC507.627010
antazoline hydrochlorideHomo sapiens (human)EC504.308010
proroxan hydrochlorideHomo sapiens (human)EC500.236420
fenoldopam mesylateHomo sapiens (human)EC502.703010
formetamideHomo sapiens (human)EC500.576210
antazoline phosphateHomo sapiens (human)EC509.970010
sercHomo sapiens (human)EC501.245010
8-anilino-1,3-dimethyl-7H-purine-2,6-dioneHomo sapiens (human)EC505.668010
N-[3-(2-phenylethyl)-2,4-dihydro-1H-1,3,5-triazin-6-yl]-1,3-benzoxazol-2-amineHomo sapiens (human)EC502.195010
N-(2-fluorophenyl)-4-phenylmethoxybenzamideHomo sapiens (human)EC5011.408010
4-[5-(2-phenylethyl)-2-sulfanylidene-1,3,5-triazinan-1-yl]benzoic acid ethyl esterHomo sapiens (human)EC500.068510
N-(2-phenylethyl)-5-thiophen-2-yl-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamideHomo sapiens (human)EC500.346210
N1-phenethylhydrazine-1-carbothioamideHomo sapiens (human)EC500.667110
phenacylamine monohydrochlorideHomo sapiens (human)EC501.078010
(1R,2S)-tranylcypromine hydrochlorideHomo sapiens (human)EC500.611010
2,6-difluoro-N-[2-[3-[(2-fluorophenyl)methylthio]-1-indolyl]ethyl]benzamideHomo sapiens (human)EC5029.913020
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[5-methyl-2-(4-methylphenyl)-4-oxazolyl]methylsulfonyl]ethanoneHomo sapiens (human)EC502.230010
guanabenzHomo sapiens (human)EC503.327010
3-methoxytyramine hydrochlorideHomo sapiens (human)EC502.402010
1-hydroxy-5-nitro-N-(2-phenylethyl)-4-spiro[benzimidazole-2,1'-cyclohexane]imineHomo sapiens (human)EC503.091010