Page last updated: 2024-09-03

pd 145065 and cocaine

pd 145065 has been researched along with cocaine in 2 studies

Compound Research Comparison

Studies
(pd 145065)
Trials
(pd 145065)
Recent Studies (post-2010)
(pd 145065)
Studies
(cocaine)
Trials
(cocaine)
Recent Studies (post-2010) (cocaine)
761532,4611,0969,400

Protein Interaction Comparison

ProteinTaxonomypd 145065 (IC50)cocaine (IC50)
Amyloid-beta precursor proteinHomo sapiens (human)0.338
Fatty acid-binding protein, heartHomo sapiens (human)0.367
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0855
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0855
DRattus norvegicus (Norway rat)5.7544
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)5.7544
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.2861
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.4321
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0855
Sodium-dependent serotonin transporterHomo sapiens (human)0.5442
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.8885
Sodium-dependent dopamine transporter Homo sapiens (human)0.3796
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.541
Sodium-dependent dopamine transporterMus musculus (house mouse)0.2
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.05
TransporterRattus norvegicus (Norway rat)3.2277

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fandino, J; Rapoport, RM; Sherman, JD; Zuccarello, M1
Rapoport, RM; Yoon, S; Zuccarello, M1

Other Studies

2 other study(ies) available for pd 145065 and cocaine

ArticleYear
Cocaine-induced endothelin-1-dependent spasm in rabbit basilar artery in vivo.
    Journal of cardiovascular pharmacology, 2003, Volume: 41, Issue:2

    Topics: Animals; Basilar Artery; Cocaine; Dose-Response Relationship, Drug; Endothelin Receptor Antagonists; Endothelin-1; Male; Oligopeptides; Rabbits; Receptor, Endothelin A; Receptors, Endothelin; Vasoconstriction

2003
Cocaine constriction of rat basilar artery in situ: roles of nitric oxide and endothelin-1.
    Pharmacology, 2014, Volume: 93, Issue:3-4

    Topics: Animals; Basilar Artery; Capsaicin; Cocaine; Dose-Response Relationship, Drug; Endothelin-1; Male; Nitric Oxide; Nitric Oxide Synthase; Oligopeptides; Rats; Rats, Sprague-Dawley; Vasoconstriction

2014