Page last updated: 2024-09-03

indatraline and cocaine

indatraline has been researched along with cocaine in 6 studies

Compound Research Comparison

Studies
(indatraline)
Trials
(indatraline)
Recent Studies (post-2010)
(indatraline)
Studies
(cocaine)
Trials
(cocaine)
Recent Studies (post-2010) (cocaine)
4602432,4611,0969,400

Protein Interaction Comparison

ProteinTaxonomyindatraline (IC50)cocaine (IC50)
Amyloid-beta precursor proteinHomo sapiens (human)0.338
Fatty acid-binding protein, heartHomo sapiens (human)0.367
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0855
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0855
DRattus norvegicus (Norway rat)5.7544
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)5.7544
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.2861
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.4321
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0855
Sodium-dependent serotonin transporterHomo sapiens (human)0.5442
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.8885
Sodium-dependent dopamine transporter Homo sapiens (human)0.3796
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.541
Sodium-dependent dopamine transporterMus musculus (house mouse)0.2
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.05
TransporterRattus norvegicus (Norway rat)3.2277

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (50.00)18.2507
2000's3 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Froimowitz, M; Gardner, EL; George, C; Haidar, RM; Jurayj, J; Moussa, A; Wu, KM1
Bergman, J; Madras, BK; Rosenzweig-Lipson, S; Spealman, RD1
al-Tikriti, MS; Baldwin, RM; Laruelle, M; Malison, RT; Neumeyer, JL; Sybirska, EH; Wisniewski, G; Zea-Ponce, Y; Zimmermann, RC; Zoghbi, SS1
Brandt, MR; Mello, NK; Negus, SS1
Mello, NK; Negus, SS1
Schenk, S1

Other Studies

6 other study(ies) available for indatraline and cocaine

ArticleYear
Slow-onset, long-duration 3-(3',4'-dichlorophenyl)-1-indanamine monoamine reuptake blockers as potential medications to treat cocaine abuse.
    Journal of medicinal chemistry, 2000, Dec-28, Volume: 43, Issue:26

    Topics: Animals; Carrier Proteins; Cell Line; Cloning, Molecular; Cocaine-Related Disorders; Crystallography, X-Ray; Discrimination Learning; Dopamine; Dopamine Plasma Membrane Transport Proteins; Humans; Indans; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Motor Activity; Nerve Tissue Proteins; Neurotransmitter Uptake Inhibitors; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Plasma Membrane Transport Proteins; Stereoisomerism; Structure-Activity Relationship; Symporters

2000
Stereoselective behavioral effects of Lu 19-005 in monkeys: relation to binding at cocaine recognition sites.
    Psychopharmacology, 1992, Volume: 107, Issue:2-3

    Topics: Animals; Behavior, Animal; Binding, Competitive; Carrier Proteins; Cocaine; Conditioning, Operant; Dopamine; Indans; Ligands; Male; Piperazines; Receptors, Drug; Reinforcement Schedule; Saimiri; Stereoisomerism

1992
SPECT imaging of dopamine and serotonin transporters with [123I]beta-CIT: pharmacological characterization of brain uptake in nonhuman primates.
    Synapse (New York, N.Y.), 1993, Volume: 13, Issue:4

    Topics: Animals; Brain; Brain Chemistry; Carrier Proteins; Chlorocebus aethiops; Citalopram; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Indans; Iodine Radioisotopes; Levodopa; Ligands; Maprotiline; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurotransmitter Uptake Inhibitors; Papio; Piperazines; Selective Serotonin Reuptake Inhibitors; Serotonin Plasma Membrane Transport Proteins; Tomography, Emission-Computed, Single-Photon

1993
Effects of the long-acting monoamine reuptake inhibitor indatraline on cocaine self-administration in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:1

    Topics: Animals; Body Weight; Cocaine; Cocaine-Related Disorders; Discrimination Learning; Dopamine Uptake Inhibitors; Indans; Macaca mulatta; Psychomotor Performance; Reinforcement, Psychology; Self Administration

1999
Effects of indatraline and buprenorphine on self-administration of speedball combinations of cocaine and heroin by rhesus monkeys.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2001, Volume: 25, Issue:1

    Topics: Animals; Buprenorphine; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Combinations; Drug Interactions; Female; Heroin; Heroin Dependence; Indans; Macaca mulatta; Male; Methylamines; Narcotics; Neurotransmitter Uptake Inhibitors; Self Administration

2001
Effects of GBR 12909, WIN 35,428 and indatraline on cocaine self-administration and cocaine seeking in rats.
    Psychopharmacology, 2002, Volume: 160, Issue:3

    Topics: Animals; Behavior, Addictive; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Indans; Male; Methylamines; Neurotransmitter Uptake Inhibitors; Piperazines; Rats; Rats, Sprague-Dawley; Self Administration

2002