gbr 13069 has been researched along with cocaine in 2 studies
Studies (gbr 13069) | Trials (gbr 13069) | Recent Studies (post-2010) (gbr 13069) | Studies (cocaine) | Trials (cocaine) | Recent Studies (post-2010) (cocaine) |
---|---|---|---|---|---|
6 | 0 | 0 | 32,461 | 1,096 | 9,400 |
Protein | Taxonomy | gbr 13069 (IC50) | cocaine (IC50) |
---|---|---|---|
Amyloid-beta precursor protein | Homo sapiens (human) | 0.338 | |
Fatty acid-binding protein, heart | Homo sapiens (human) | 0.367 | |
5-hydroxytryptamine receptor 2C | Rattus norvegicus (Norway rat) | 0.0855 | |
5-hydroxytryptamine receptor 2A | Rattus norvegicus (Norway rat) | 0.0855 | |
D | Rattus norvegicus (Norway rat) | 5.7544 | |
Alpha-2B adrenergic receptor | Rattus norvegicus (Norway rat) | 5.7544 | |
Alpha-2C adrenergic receptor | Rattus norvegicus (Norway rat) | 5.7544 | |
Alpha-2A adrenergic receptor | Rattus norvegicus (Norway rat) | 5.7544 | |
Sodium-dependent noradrenaline transporter | Homo sapiens (human) | 1.2861 | |
Sodium-dependent dopamine transporter | Rattus norvegicus (Norway rat) | 0.4321 | |
5-hydroxytryptamine receptor 2B | Rattus norvegicus (Norway rat) | 0.0855 | |
Sodium-dependent serotonin transporter | Homo sapiens (human) | 0.5442 | |
Sodium-dependent serotonin transporter | Rattus norvegicus (Norway rat) | 0.8885 | |
Sodium-dependent dopamine transporter | Homo sapiens (human) | 0.3796 | |
Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | 5.541 | |
Sodium-dependent dopamine transporter | Mus musculus (house mouse) | 0.2 | |
Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | 1.05 | |
Transporter | Rattus norvegicus (Norway rat) | 3.2277 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (50.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Grundt, P; Katz, JL; Kopajtic, T; Kulkarni, SS; Newman, AH | 1 |
Heikkila, RE; Kindt, MV; Mayer, RA | 1 |
2 other study(ies) available for gbr 13069 and cocaine
Article | Year |
---|---|
Structure-activity relationships at monoamine transporters for a series of N-substituted 3alpha-(bis[4-fluorophenyl]methoxy)tropanes: comparative molecular field analysis, synthesis, and pharmacological evaluation.
Topics: Animals; Brain; Carrier Proteins; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; In Vitro Techniques; Male; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Nerve Tissue Proteins; Norepinephrine Plasma Membrane Transport Proteins; Protein Binding; Quantitative Structure-Activity Relationship; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Serotonin Plasma Membrane Transport Proteins; Symporters; Tropanes | 2004 |
Prevention of the nigrostriatal toxicity of 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine by inhibitors of 3,4-dihydroxyphenylethylamine transport.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 1-Methyl-4-phenylpyridinium; Animals; Biological Transport; Cocaine; Corpus Striatum; Dopamine; Dopamine Antagonists; Flunarizine; Male; Mice; Nalidixic Acid; Naphthyridines; Piperazines; Pyridines; Pyridinium Compounds; Pyrroles; Rats; Rats, Inbred Strains; Substantia Nigra | 1986 |