Page last updated: 2024-09-03

aj 76 and cocaine

aj 76 has been researched along with cocaine in 5 studies

Compound Research Comparison

Studies
(aj 76)
Trials
(aj 76)
Recent Studies (post-2010)
(aj 76)
Studies
(cocaine)
Trials
(cocaine)
Recent Studies (post-2010) (cocaine)
370232,4611,0969,400

Protein Interaction Comparison

ProteinTaxonomyaj 76 (IC50)cocaine (IC50)
Amyloid-beta precursor proteinHomo sapiens (human)0.338
Fatty acid-binding protein, heartHomo sapiens (human)0.367
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0855
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0855
DRattus norvegicus (Norway rat)5.7544
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)5.7544
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.2861
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.4321
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0855
Sodium-dependent serotonin transporterHomo sapiens (human)0.5442
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.8885
Sodium-dependent dopamine transporter Homo sapiens (human)0.3796
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.541
Sodium-dependent dopamine transporterMus musculus (house mouse)0.2
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.05
TransporterRattus norvegicus (Norway rat)3.2277

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carlsson, A; Hoffmann, WE; Ljung, E; Lum, JT; Piercey, MF; Svensson, K1
Callahan, PM; Cunningham, KA; Piercey, MF1
Piercey, MF; Vanover, KE; Woolverton, WL1
Collins, RJ; Myers, JE; Piercey, MF; Richardson, NR; Roberts, DC; Svensson, K1
Casey, BL; Piercey, MF; Ray, CA1

Other Studies

5 other study(ies) available for aj 76 and cocaine

ArticleYear
Antagonism of cocaine's pharmacological effects by the stimulant dopaminergic antagonists, (+)-AJ76 and (+)-UH232.
    Brain research, 1992, Aug-21, Volume: 588, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Brain Chemistry; Cocaine; Dihydroxyphenylalanine; Dopamine; Dopamine Antagonists; Electrophysiology; Homovanillic Acid; Male; Microelectrodes; Motor Activity; Rats; Rats, Sprague-Dawley; Tetrahydronaphthalenes

1992
Effects of the putative dopamine autoreceptor antagonists (+)-AJ 76 and (+)-UH 232 on the discriminative stimulus properties of cocaine.
    Psychopharmacology, 1992, Volume: 107, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Cocaine; Discrimination, Psychological; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Male; Rats; Rats, Inbred Strains; Tetrahydronaphthalenes

1992
Evaluation of the reinforcing and discriminative stimulus effects of cocaine in combination with (+)-AJ76 or clozapine.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:2

    Topics: Animals; Clozapine; Cocaine; Discrimination Learning; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Macaca mulatta; Male; Reinforcement, Psychology; Tetrahydronaphthalenes

1993
Antagonism of cocaine self-administration by the preferential dopamine autoreceptor antagonist, (+)-AJ 76.
    Brain research, 1993, Aug-13, Volume: 619, Issue:1-2

    Topics: Animals; Cocaine; Conditioning, Operant; Dextroamphetamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Male; Rats; Rats, Sprague-Dawley; Self Administration; Stereoisomerism; Substance-Related Disorders; Tetrahydronaphthalenes

1993
Antagonism of cocaine's stimulant effects on local cerebral glucose utilization by the preferential autoreceptor antagonist (+)-AJ 76.
    Journal of neural transmission (Vienna, Austria : 1996), 1996, Volume: 103, Issue:3

    Topics: Animals; Autoradiography; Autoreceptors; Brain Chemistry; Central Nervous System Stimulants; Cocaine; Deoxyglucose; Dopamine Antagonists; Energy Metabolism; Glucose; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Tetrahydronaphthalenes

1996