| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| activating transcription factor 6 | Homo sapiens (human) | Potency | 24.5412 | 1 | 1 |
| apical membrane antigen 1, AMA1 | Plasmodium falciparum 3D7 | Potency | 28.1838 | 1 | 1 |
| AR protein | Homo sapiens (human) | Potency | 36.9017 | 9 | 13 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 30.9100 | 3 | 3 |
| bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 11.2202 | 1 | 1 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 48.2037 | 1 | 4 |
| Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 53.1764 | 1 | 2 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 5.6234 | 1 | 1 |
| chromobox protein homolog 1 | Homo sapiens (human) | Potency | 78.1614 | 1 | 3 |
| cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 15.4871 | 1 | 1 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 7.7619 | 1 | 1 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 27.3060 | 1 | 1 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 47.0145 | 9 | 13 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 30.6379 | 1 | 1 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 29.1048 | 5 | 6 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 24.0759 | 1 | 3 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 25.4241 | 2 | 2 |
| G | Vesicular stomatitis virus | Potency | 15.4871 | 1 | 1 |
| geminin | Homo sapiens (human) | Potency | 22.2368 | 2 | 3 |
| GLI family zinc finger 3 | Homo sapiens (human) | Potency | 68.5896 | 2 | 2 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 18.0147 | 2 | 3 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 61.1306 | 1 | 1 |
| heat shock protein beta-1 | Homo sapiens (human) | Potency | 6.2555 | 1 | 2 |
| histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 35.4813 | 1 | 1 |
| HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 15.4871 | 1 | 1 |
| hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 43.6412 | 1 | 1 |
| Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 15.4871 | 1 | 2 |
| Interferon beta | Homo sapiens (human) | Potency | 15.4871 | 1 | 1 |
| lamin isoform A-delta10 | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
| lethal(3)malignant brain tumor-like protein 1 isoform I | Homo sapiens (human) | Potency | 14.1254 | 1 | 1 |
| Luciferase | Photinus pyralis (common eastern firefly) | Potency | 28.6402 | 2 | 2 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 44.2357 | 4 | 7 |
| nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 29.0929 | 1 | 1 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 30.8956 | 1 | 1 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 35.4813 | 1 | 1 |
| nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 22.5981 | 3 | 10 |
| parathyroid hormone/parathyroid hormone-related peptide receptor precursor | Homo sapiens (human) | Potency | 15.1652 | 1 | 2 |
| peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | Potency | 100.0000 | 1 | 1 |
| peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 14.3818 | 1 | 1 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 44.9815 | 2 | 3 |
| phosphopantetheinyl transferase | Bacillus subtilis | Potency | 39.8107 | 1 | 1 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 31.1924 | 2 | 7 |
| pregnane X receptor | Rattus norvegicus (Norway rat) | Potency | 37.2750 | 1 | 4 |
| progesterone receptor | Homo sapiens (human) | Potency | 54.4827 | 1 | 1 |
| RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 55.6553 | 2 | 4 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 56.7390 | 3 | 4 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 20.2782 | 3 | 7 |
| serine-protein kinase ATM isoform a | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Potency | 23.7781 | 1 | 1 |
| TDP1 protein | Homo sapiens (human) | Potency | 13.2780 | 2 | 2 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 68.5896 | 2 | 2 |
| thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 0.0052 | 1 | 2 |
| thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 26.6448 | 3 | 3 |
| USP1 protein, partial | Homo sapiens (human) | Potency | 50.1187 | 1 | 1 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 43.6412 | 1 | 1 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 28.0740 | 3 | 4 |
| vitamin D3 receptor isoform VDRA | Homo sapiens (human) | Potency | 75.0594 | 1 | 2 |
| Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 61.1306 | 1 | 1 |