Page last updated: 2024-09-05

sb 216763 and ag 1879

sb 216763 has been researched along with ag 1879 in 2 studies

Compound Research Comparison

Studies
(sb 216763)
Trials
(sb 216763)
Recent Studies (post-2010)
(sb 216763)
Studies
(ag 1879)
Trials
(ag 1879)
Recent Studies (post-2010) (ag 1879)
34202255750215

Protein Interaction Comparison

ProteinTaxonomysb 216763 (IC50)ag 1879 (IC50)
Chain A, Lck KinaseHomo sapiens (human)0.02
Chain A, Tyrosine-protein kinase LynMus musculus (house mouse)0.009
Chain A, Tyrosine-protein kinase LynMus musculus (house mouse)0.009
Receptor-interacting serine/threonine-protein kinase 2Homo sapiens (human)0.019
Proto-oncogene tyrosine-protein kinase SrcGallus gallus (chicken)0.036
Epidermal growth factor receptorHomo sapiens (human)0.48
Tyrosine-protein kinase LckHomo sapiens (human)0.004
Proto-oncogene tyrosine-protein kinase LCK Mus musculus (house mouse)0.031
Tyrosine-protein kinase FynHomo sapiens (human)0.0052
Tyrosine-protein kinase LynHomo sapiens (human)0.0005
Tyrosine-protein kinase HCKHomo sapiens (human)0.005
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)1.1814
Tyrosine-protein kinase CSKHomo sapiens (human)0.5
Casein kinase I isoform deltaHomo sapiens (human)0.041
Mitogen-activated protein kinase 14Homo sapiens (human)4.23

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Fujibayashi, M; Kato, S; Koriyama, Y; Takadera, T1

Other Studies

2 other study(ies) available for sb 216763 and ag 1879

ArticleYear
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
Apoptosis induced by SRC-family tyrosine kinase inhibitors in cultured rat cortical cells.
    Neurotoxicity research, 2012, Volume: 21, Issue:3

    Topics: Animals; Apoptosis; Benzazepines; Caspase 3; Caspase 9; Cells, Cultured; Cerebral Cortex; Enzyme Inhibitors; Female; Focal Adhesion Protein-Tyrosine Kinases; Glycogen Synthase Kinase 3; Indoles; Insulin-Like Growth Factor I; Maleimides; MAP Kinase Signaling System; Neurons; Neuroprotective Agents; Pregnancy; Proto-Oncogene Proteins c-akt; Pyrimidines; Rats; Rats, Wistar; src-Family Kinases; Sulfonamides

2012
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