Page last updated: 2024-09-05

piboserod and morphine

piboserod has been researched along with morphine in 3 studies

Compound Research Comparison

Studies
(piboserod)
Trials
(piboserod)
Recent Studies (post-2010)
(piboserod)
Studies
(morphine)
Trials
(morphine)
Recent Studies (post-2010) (morphine)
11955344,2705,2008,695

Protein Interaction Comparison

ProteinTaxonomypiboserod (IC50)morphine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.2939
Delta-type opioid receptorRattus norvegicus (Norway rat)0.2278
Kappa-type opioid receptorMus musculus (house mouse)0.0828
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0385
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0545
Mu-type opioid receptorHomo sapiens (human)0.122
Delta-type opioid receptorHomo sapiens (human)0.1199
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.9308
Kappa-type opioid receptorHomo sapiens (human)0.655
Mu-type opioid receptorMus musculus (house mouse)0.3305
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.202
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.25

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Boulouard, M; Bureau, R; Butt-Gueulle, S; Dauphin, F; Daveu, C; Duchatelle, P; Dumuis, A; Lelong-Boulouard, V; Lemaître, S; Lepailleur, A; Lezoualc'h, F; Pfeiffer, B; Rault, S1
Alisi, MA; Apicella, C; Capezzone de Joannon, A; Cazzolla, N; Costi, R; Cuzzucoli Crucitti, G; Di Santo, R; Furlotti, G; Garrone, B; Iacovo, A; Magarò, G; Mangano, G; Miele, G; Ombrato, R; Pescatori, L; Polenzani, L; Rosi, F; Vitiello, M1
Hayashi, SS; Kamei, J; Nakanishi, Y; Ohsawa, M1

Other Studies

3 other study(ies) available for piboserod and morphine

ArticleYear
Novel antagonists of serotonin-4 receptors: synthesis and biological evaluation of pyrrolothienopyrazines.
    Bioorganic & medicinal chemistry, 2009, Mar-15, Volume: 17, Issue:6

    Topics: Animals; Chlorocebus aethiops; COS Cells; Humans; Indoles; Models, Molecular; Molecular Structure; Pyrazines; Radioligand Assay; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sulfonamides

2009
Discovery and pharmacological profile of new 1H-indazole-3-carboxamide and 2H-pyrrolo[3,4-c]quinoline derivatives as selective serotonin 4 receptor ligands.
    Journal of medicinal chemistry, 2012, Nov-26, Volume: 55, Issue:22

    Topics: Animals; Computational Biology; Dogs; Drug Design; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Ligands; Macaca fascicularis; Mice; Microsomes, Liver; Molecular Structure; Nociception; Protein Binding; Quinolines; Radioligand Assay; Rats; Receptors, Serotonin, 5-HT4; Structure-Activity Relationship; Swine

2012
Effect of chronic pain on morphine-induced respiratory depression in mice.
    Neuroscience, 2011, Feb-03, Volume: 174

    Topics: Analgesics, Opioid; Animals; Benzamides; Brain Stem; Chronic Disease; Indoles; Ligation; Male; Mice; Mice, Inbred ICR; Morphine; Morpholines; Pain; Peripheral Nervous System Diseases; Receptors, Serotonin, 5-HT4; Respiration; Respiratory Insufficiency; Sciatic Nerve; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides

2011