Page last updated: 2024-09-02

npc 12626 and naloxone

npc 12626 has been researched along with naloxone in 6 studies

Compound Research Comparison

Studies
(npc 12626)
Trials
(npc 12626)
Recent Studies (post-2010)
(npc 12626)
Studies
(naloxone)
Trials
(naloxone)
Recent Studies (post-2010) (naloxone)
550020,1341,2573,321

Protein Interaction Comparison

ProteinTaxonomynpc 12626 (IC50)naloxone (IC50)
Cytochrome P450 2D6Homo sapiens (human)2
Delta-type opioid receptorMus musculus (house mouse)0.043
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0219
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0019
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0019
Mu-type opioid receptorHomo sapiens (human)0.0397
Delta-type opioid receptorHomo sapiens (human)0.1896
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.05
Kappa-type opioid receptorHomo sapiens (human)0.0795
Mu-type opioid receptorMus musculus (house mouse)0.0154
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0089
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.0055

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (83.33)18.2507
2000's1 (16.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kavaliers, M; Saucier, DM1
Popik, P; Skolnick, P1
Colwell, DD; Kavaliers, M; Perrot-Sinal, TS1
Choleris, E; Colwell, DD; Kavaliers, M3

Other Studies

6 other study(ies) available for npc 12626 and naloxone

ArticleYear
Antagonistic effects of the selective, competitive N-methyl-D-aspartate (NMDA) receptor antagonist, NPC 12626, on kappa opiate-induced analgesia in male deer mice.
    Brain research, 1994, Feb-21, Volume: 637, Issue:1-2

    Topics: Amino Acids; Analgesics; Animals; Benzeneacetamides; Dizocilpine Maleate; Dose-Response Relationship, Drug; Male; Morphine; Naloxone; Naltrexone; Nociceptors; Pain Measurement; Peromyscus; Pyrrolidines; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa

1994
The NMDA antagonist memantine blocks the expression and maintenance of morphine dependence.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:4

    Topics: Amino Acids; Animals; Brain Chemistry; Dose-Response Relationship, Drug; Electrophysiology; Excitatory Amino Acid Antagonists; Glycine; Male; Memantine; Mice; Morphine Dependence; Motor Activity; Naloxone; Narcotic Antagonists; Receptors, N-Methyl-D-Aspartate

1996
Opioid and non-opioid NMDA-mediated predator-induced analgesia in mice and the effects of parasitic infection.
    Brain research, 1997, Aug-22, Volume: 766, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amino Acids; Analgesia; Animals; Behavior, Animal; Bicuculline; Butyrates; Butyric Acid; Excitatory Amino Acid Antagonists; GABA Antagonists; Histamine Antagonists; Host-Parasite Interactions; Male; Mice; Mice, Inbred Strains; Naloxone; Narcotic Antagonists; Nematospiroides dubius; Nociceptors; Odorants; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Serotonin Receptor Agonists; Stress, Physiological; Strongylida Infections; Time Factors

1997
Analgesic responses of male mice exposed to the odors of parasitized females: effects of male sexual experience and infection status.
    Behavioral neuroscience, 1998, Volume: 112, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amino Acids; Analgesia; Analysis of Variance; Animals; Choice Behavior; Discrimination, Psychological; Estrus; Excitatory Amino Acid Antagonists; Female; Male; Mice; Mice, Inbred Strains; Naloxone; Narcotic Antagonists; Nematospiroides dubius; Odorants; Pain Threshold; Practice, Psychological; Serotonin Receptor Agonists; Sexual Behavior, Animal; Smell; Stress, Psychological; Strongylida Infections; Time Factors

1998
Sex differences in opioid and N-methyl-D-aspartate mediated non-opioid biting fly exposure induced analgesia in deer mice.
    Pain, 1998, Volume: 77, Issue:2

    Topics: Amino Acids; Analgesia; Analysis of Variance; Animals; Behavior, Animal; Excitatory Amino Acid Antagonists; Female; Houseflies; Insect Bites and Stings; Male; Naloxone; Naltrexone; Narcotic Antagonists; Nociceptors; Peromyscus; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa; Sex Characteristics; Stress, Physiological

1998
NMDA-mediated social learning of fear-induced conditioned analgesia to biting flies.
    Neuroreport, 2001, Mar-26, Volume: 12, Issue:4

    Topics: Amino Acids; Analgesia; Animals; Avoidance Learning; Bites and Stings; Conditioning, Psychological; Diptera; Excitatory Amino Acid Antagonists; Fear; Male; Mice; Mice, Inbred Strains; Naloxone; Narcotic Antagonists; Nociceptors; Receptors, N-Methyl-D-Aspartate; Social Behavior

2001