Page last updated: 2024-09-03

mosapride and morphine

mosapride has been researched along with morphine in 6 studies

Compound Research Comparison

Studies
(mosapride)
Trials
(mosapride)
Recent Studies (post-2010)
(mosapride)
Studies
(morphine)
Trials
(morphine)
Recent Studies (post-2010) (morphine)
2869014244,2705,2008,695

Protein Interaction Comparison

ProteinTaxonomymosapride (IC50)morphine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.2939
Delta-type opioid receptorRattus norvegicus (Norway rat)0.2278
Kappa-type opioid receptorMus musculus (house mouse)0.0828
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0385
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0545
Mu-type opioid receptorHomo sapiens (human)0.122
Delta-type opioid receptorHomo sapiens (human)0.1199
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.9308
Kappa-type opioid receptorHomo sapiens (human)0.655
Mu-type opioid receptorMus musculus (house mouse)0.3305
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.202
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.25

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (83.33)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dkhar, SA; Shashindran, CH; Shewade, DG; Suchitra, AD1
Geisslinger, G; Hummel, T; Lötsch, J; Schneider, A; Skarke, C1
Dkhar, SA; Krishna, PR; Ramaswamy, S; Sandhiya, S1
Horie, S; Kimura, H; Matsumoto, K; Tashima, K; Uchida, M1
He, QY; Lin, HS; Zhang, FL1
Hayashi, SS; Kamei, J; Nakanishi, Y; Ohsawa, M1

Trials

2 trial(s) available for mosapride and morphine

ArticleYear
The 5-hydroxytryptamine 4 receptor agonist mosapride does not antagonize morphine-induced respiratory depression.
    Clinical pharmacology and therapeutics, 2005, Volume: 78, Issue:3

    Topics: Adult; Analgesics, Opioid; Animals; Benzamides; Carbon Dioxide; Cross-Over Studies; Double-Blind Method; Female; Humans; Male; Morphine; Morpholines; Naloxone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT4; Respiratory Insufficiency; Serotonin Receptor Agonists

2005
[Effect of electro-acupuncture in treating morphine sulfate caused constipation in tumor patients].
    Zhongguo Zhong xi yi jie he za zhi Zhongguo Zhongxiyi jiehe zazhi = Chinese journal of integrated traditional and Western medicine, 2009, Volume: 29, Issue:10

    Topics: Adult; Aged; Aged, 80 and over; Benzamides; Constipation; Electroacupuncture; Female; Humans; Male; Middle Aged; Morphine; Morpholines; Neoplasms

2009

Other Studies

4 other study(ies) available for mosapride and morphine

ArticleYear
Relative efficacy of some prokinetic drugs in morphine-induced gastrointestinal transit delay in mice.
    World journal of gastroenterology, 2003, Volume: 9, Issue:4

    Topics: Animals; Benzamides; Cisapride; Domperidone; Drug Interactions; Erythromycin; Female; Gastric Emptying; Gastrointestinal Transit; Male; Metoclopramide; Mice; Morphine; Morpholines

2003
Role of ion channel modifiers in reversal of morphine-induced gastrointestinal inertia by prokinetic agents in mice.
    Indian journal of experimental biology, 2008, Volume: 46, Issue:1

    Topics: Analgesics, Opioid; Animals; Benzamides; Calcium Channels; Domperidone; Gastrointestinal Tract; Glyburide; Intestine, Small; Ion Channels; Kinetics; Mice; Minoxidil; Morphine; Morpholines; Nifedipine; Time Factors

2008
Validation of 13C-acetic acid breath test by measuring effects of loperamide, morphine, mosapride, and itopride on gastric emptying in mice.
    Biological & pharmaceutical bulletin, 2008, Volume: 31, Issue:10

    Topics: Acetic Acid; Analgesics, Opioid; Animals; Anti-Ulcer Agents; Antidiarrheals; Antiemetics; Benzamides; Benzyl Compounds; Breath Tests; Coloring Agents; Gastric Emptying; Loperamide; Male; Mice; Morphine; Morpholines; Naloxone; Narcotic Antagonists; Phenolsulfonphthalein; Reproducibility of Results

2008
Effect of chronic pain on morphine-induced respiratory depression in mice.
    Neuroscience, 2011, Feb-03, Volume: 174

    Topics: Analgesics, Opioid; Animals; Benzamides; Brain Stem; Chronic Disease; Indoles; Ligation; Male; Mice; Mice, Inbred ICR; Morphine; Morpholines; Pain; Peripheral Nervous System Diseases; Receptors, Serotonin, 5-HT4; Respiration; Respiratory Insufficiency; Sciatic Nerve; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides

2011
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