Page last updated: 2024-08-07 15:40:58

Muscarinic acetylcholine receptor M2

A muscarinic acetylcholine receptor M2 that is encoded in the genome of pig. [OMA:P06199, PRO:DNx]

Synonyms

Research

Bioassay Publications (9)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's1 (11.11)18.2507
2000's7 (77.78)29.6817
2010's1 (11.11)24.3611
2020's0 (0.00)2.80

Compounds (13)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
cocaineSus scrofa (pig)Ki0.234411
pd 168,077Sus scrofa (pig)Ki0.017011
3-[bis(4-fluorophenyl)methoxy]-8-methyl-8-azabicyclo[3.2.1]octaneSus scrofa (pig)Ki0.013811

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
tacrineSus scrofa (pig)EC506.304812
verapamilSus scrofa (pig)EC5030.974211
gallamine triethiodideSus scrofa (pig)EC500.130912
methoctramineSus scrofa (pig)EC502.999211
hexamethylenebis(dimethyl-(3-phthalimidopropyl)ammonium bromide)Sus scrofa (pig)EC501.053744
w 84Sus scrofa (pig)EC501.438811
heptane-1,7-bis(dimethyl-3'-phthalimidopropylammonium)Sus scrofa (pig)EC500.389011
caracurine vSus scrofa (pig)EC500.436011
jnj-5207852Sus scrofa (pig)Kd0.000111
thioperamideSus scrofa (pig)Kd0.043611