Page last updated: 2024-09-03

tifluadom and nalorphine

tifluadom has been researched along with nalorphine in 3 studies

Compound Research Comparison

Studies
(tifluadom)
Trials
(tifluadom)
Recent Studies (post-2010)
(tifluadom)
Studies
(nalorphine)
Trials
(nalorphine)
Recent Studies (post-2010) (nalorphine)
78001,134416

Protein Interaction Comparison

ProteinTaxonomytifluadom (IC50)nalorphine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.1095
Delta-type opioid receptorRattus norvegicus (Norway rat)0.004
Kappa-type opioid receptorMus musculus (house mouse)0.1095
Mu-type opioid receptorRattus norvegicus (Norway rat)0.004
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.004
Mu-type opioid receptorMus musculus (house mouse)0.1095
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.006

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19902 (66.67)18.7374
1990's1 (33.33)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, C; Li, JG; Liu-Chen, LY; Luo, LY; Zhu, J1
Hayes, A; Kelly, A1
Code, RA; Tang, AH1

Other Studies

3 other study(ies) available for tifluadom and nalorphine

ArticleYear
Activation of the cloned human kappa opioid receptor by agonists enhances [35S]GTPgammaS binding to membranes: determination of potencies and efficacies of ligands.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylate Cyclase Toxin; Animals; Binding Sites; Cell Membrane; CHO Cells; Cholera Toxin; Cloning, Molecular; Cricetinae; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Humans; Kinetics; Magnesium; Pertussis Toxin; Pyrrolidines; Receptors, Opioid, kappa; Recombinant Proteins; Sodium; Sulfur Radioisotopes; Virulence Factors, Bordetella

1997
Profile of activity of kappa receptor agonists in the rabbit vas deferens.
    European journal of pharmacology, 1985, Apr-16, Volume: 110, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Cyclazocine; Ethylketocyclazocine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nalorphine; Naloxone; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens

1985
Discriminative stimulus properties of nalorphine in the rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:3

    Topics: Animals; Benzodiazepines; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Macaca mulatta; Male; Nalorphine; Naloxone; Phenazocine; Receptors, Opioid; Receptors, Opioid, kappa

1983