Page last updated: 2024-09-03

cki 7 and h 89

cki 7 has been researched along with h 89 in 3 studies

Compound Research Comparison

Studies
(cki 7)
Trials
(cki 7)
Recent Studies (post-2010)
(cki 7)
Studies
(h 89)
Trials
(h 89)
Recent Studies (post-2010) (h 89)
35071,6190409

Protein Interaction Comparison

ProteinTaxonomycki 7 (IC50)h 89 (IC50)
Rho-associated protein kinase 2Homo sapiens (human)1.9504
Ribosomal protein S6 kinase alpha-5Homo sapiens (human)0.12
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)0.073
cAMP-dependent protein kinase catalytic subunit alpha Mus musculus (house mouse)0.381
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)0.6365
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)0.6365
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)0.6365
Ribosomal protein S6 kinase beta-1Homo sapiens (human)0.08
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)1.9886
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)0.5417
Rho-associated protein kinase 2Rattus norvegicus (Norway rat)0.27
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)0.3207

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Hidaka, H; Kobayashi, R; Watanabe, M1
Hidaka, H; Kobayashi, R1

Reviews

1 review(s) available for cki 7 and h 89

ArticleYear
[Molecular pharmacology of intracellular calcium signaling].
    Seikagaku. The Journal of Japanese Biochemical Society, 1990, Volume: 62, Issue:12

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Azepines; Calcium; Cyclic AMP; Humans; Isoquinolines; Muscle Contraction; Muscle, Smooth; Myosins; Phosphorylation; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Second Messenger Systems; Sulfonamides

1990

Other Studies

2 other study(ies) available for cki 7 and h 89

ArticleYear
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
Properties and use of H-series compounds as protein kinase inhibitors.
    Methods in enzymology, 1991, Volume: 201

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Casein Kinases; Isoquinolines; Kinetics; PC12 Cells; Piperazines; Protein Binding; Protein Kinase Inhibitors; Protein Kinases; Sulfonamides

1991