Page last updated: 2024-09-05

ag 112 and ag-213

ag 112 has been researched along with ag-213 in 4 studies

Compound Research Comparison

Studies
(ag 112)
Trials
(ag 112)
Recent Studies (post-2010)
(ag 112)
Studies
(ag-213)
Trials
(ag-213)
Recent Studies (post-2010) (ag-213)
1901022404

Protein Interaction Comparison

ProteinTaxonomyag 112 (IC50)ag-213 (IC50)
Epidermal growth factor receptorHomo sapiens (human)3.222
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)5.7
Macrophage colony-stimulating factor 1 receptorHomo sapiens (human)3.0667
Protein kinase C alpha typeHomo sapiens (human)3
Protein-glutamine gamma-glutamyltransferase 2Homo sapiens (human)3
M-phase inducer phosphatase 1Homo sapiens (human)3
Tyrosine-protein kinase JAK3Homo sapiens (human)3
Receptor-type tyrosine-protein phosphatase etaHomo sapiens (human)3
Receptor protein-tyrosine kinase Homo sapiens (human)3

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19901 (25.00)18.7374
1990's1 (25.00)18.2507
2000's2 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chang, CJ; Geahlen, RL1
Gazit, A; Gilon, C; Levitzki, A; Yaish, P1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1

Reviews

1 review(s) available for ag 112 and ag-213

ArticleYear
Protein-tyrosine kinase inhibition: mechanism-based discovery of antitumor agents.
    Journal of natural products, 1992, Volume: 55, Issue:11

    Topics: Animals; Antineoplastic Agents; Drug Screening Assays, Antitumor; Humans; Protein-Tyrosine Kinases

1992

Other Studies

3 other study(ies) available for ag 112 and ag-213

ArticleYear
Tyrphostins I: synthesis and biological activity of protein tyrosine kinase inhibitors.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:10

    Topics: Benzylidene Compounds; Carcinoma, Squamous Cell; Cell Division; Cell Line; Epidermal Growth Factor; ErbB Receptors; Humans; Kinetics; Molecular Structure; Nitriles; Phosphorylation; Protein-Tyrosine Kinases; Structure-Activity Relationship

1989
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009