Page last updated: 2024-08-07 13:50:31
Glutamate receptor 4
A glutamate receptor 4 that is encoded in the genome of mouse. [OMA:Q9Z2W8, PRO:DNx]
Synonyms
GluR-4;
GluR4;
AMPA-selective glutamate receptor 4;
GluR-D;
Glutamate receptor ionotropic, AMPA 4;
GluA4
Research
Bioassay Publications (3)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (33.33) | 18.2507 |
2000's | 2 (66.67) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (8)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid | Mus musculus (house mouse) | IC50 | 0.0400 | 1 | 1 |
quisqualic acid | Mus musculus (house mouse) | IC50 | 0.0800 | 1 | 1 |
4-bromohomoibotenic acid, (rs)-isomer | Mus musculus (house mouse) | IC50 | 0.6000 | 1 | 1 |
4-bromohomoibotenic acid | Mus musculus (house mouse) | IC50 | 32.0000 | 1 | 1 |
tqx 173 | Mus musculus (house mouse) | IC50 | 2.3000 | 1 | 1 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
gyki 52466 | Mus musculus (house mouse) | ED50 | 30.5500 | 2 | 2 |
cfm 2 | Mus musculus (house mouse) | ED50 | 13.8000 | 2 | 2 |
4,5-dihydro-7,8-dimethoxy-1-phenyl-3h-2,3-benzodiazepin-4-one | Mus musculus (house mouse) | ED50 | 32.8500 | 2 | 2 |