Page last updated: 2024-08-07 21:30:00

Beta-lactamase

[no definition available]

Synonyms

Research

Bioassay Publications (1)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Compounds (14)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
benzoic acidKlebsiella pneumoniaeIC502,000.000011
picolinic acidKlebsiella pneumoniaeIC502,000.000011
indolebutyric acidKlebsiella pneumoniaeIC50480.000011
biphenyl-3-carboxylic acidKlebsiella pneumoniaeIC50260.000011
4-phenylpyridineKlebsiella pneumoniaeIC502,000.000011
indole-5-carboxylic acidKlebsiella pneumoniaeIC501,390.000011
4-carboxybiphenyl etherKlebsiella pneumoniaeIC50870.000011

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
benzoic acidKlebsiella pneumoniaeKd1,000.000011
picolinic acidKlebsiella pneumoniaeKd1,000.000011
indolebutyric acidKlebsiella pneumoniaeKd430.000011
biphenyl-3-carboxylic acidKlebsiella pneumoniaeKd370.000011
4-phenylpyridineKlebsiella pneumoniaeKd1,000.000011
indole-5-carboxylic acidKlebsiella pneumoniaeKd1,380.000011
4-carboxybiphenyl etherKlebsiella pneumoniaeKd660.000011
meropenemKlebsiella pneumoniaeKd0.850011

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
penicillin gKlebsiella pneumoniaeKm700.000011
ampicillinKlebsiella pneumoniaeKm150.000011
imipenem, anhydrousKlebsiella pneumoniaeKm7.900011
centaKlebsiella pneumoniaeKm24.000011
meropenemKlebsiella pneumoniaeKm1.000011
cefepimeKlebsiella pneumoniaeKm300.000011
nitrocefinKlebsiella pneumoniaeKm120.000022