Page last updated: 2024-08-07 21:13:17
Solute carrier organic anion transporter family member 2A1
A solute carrier organic anion transporter family member 2A1 that is encoded in the genome of rat. [OMA:Q00910, PRO:DNx]
Synonyms
Matrin F/G 1;
Prostaglandin transporter;
PGT;
Solute carrier family 21 member 2
Research
Bioassay Publications (3)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (14)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
furosemide | Rattus norvegicus (Norway rat) | Ki | 47.0000 | 1 | 1 |
sulfobromophthalein sodium | Rattus norvegicus (Norway rat) | Ki | 5.8000 | 1 | 1 |
bromcresol green | Rattus norvegicus (Norway rat) | Ki | 3.6000 | 1 | 1 |
prostaglandin h2 | Rattus norvegicus (Norway rat) | Ki | 0.0382 | 1 | 1 |
prostaglandin d2 | Rattus norvegicus (Norway rat) | Ki | 0.0450 | 1 | 1 |
dinoprost | Rattus norvegicus (Norway rat) | Ki | 0.0450 | 1 | 1 |
prostaglandin b1 | Rattus norvegicus (Norway rat) | Ki | 0.0712 | 1 | 1 |
prostaglandin a1 | Rattus norvegicus (Norway rat) | Ki | 0.2860 | 1 | 1 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
arachidonic acid | Rattus norvegicus (Norway rat) | Km | 96.0000 | 1 | 1 |
dinoprostone | Rattus norvegicus (Norway rat) | Km | 0.0940 | 1 | 1 |
dinoprost | Rattus norvegicus (Norway rat) | Km | 0.1040 | 1 | 1 |
alprostadil | Rattus norvegicus (Norway rat) | Km | 0.0700 | 1 | 1 |
6-ketoprostaglandin f1 alpha | Rattus norvegicus (Norway rat) | Km | 7.5690 | 1 | 1 |
thromboxane b2 | Rattus norvegicus (Norway rat) | Km | 0.4230 | 1 | 1 |
iloprost | Rattus norvegicus (Norway rat) | Km | 86.9000 | 1 | 1 |