Page last updated: 2024-08-07 16:56:33

Melanin-concentrating hormone receptor 1

A melanin-concentrating hormone receptor 1 that is encoded in the genome of rat. [OMA:P97639, PRO:DNx]

Synonyms

MCH receptor 1;
MCH-R1;
MCHR-1;
G-protein coupled receptor 24;
MCH-1R;
MCH1R;
MCHR;
SLC-1;
Somatostatin receptor-like protein

Research

Bioassay Publications (5)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (60.00)29.6817
2010's2 (40.00)24.3611
2020's0 (0.00)2.80

Compounds (4)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
1-(3-(4-chlorobenzoyl)propyl)-4-hydroxy-4-(4-chlorophenyl)piperidineRattus norvegicus (Norway rat)Ki0.350011
gw 803430Rattus norvegicus (Norway rat)Ki0.000311
t-226296Rattus norvegicus (Norway rat)IC500.024011
snap7941Rattus norvegicus (Norway rat)Ki0.000833