Page last updated: 2024-08-07 16:56:33
Melanin-concentrating hormone receptor 1
A melanin-concentrating hormone receptor 1 that is encoded in the genome of rat. [OMA:P97639, PRO:DNx]
Synonyms
MCH receptor 1;
MCH-R1;
MCHR-1;
G-protein coupled receptor 24;
MCH-1R;
MCH1R;
MCHR;
SLC-1;
Somatostatin receptor-like protein
Research
Bioassay Publications (5)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 3 (60.00) | 29.6817 |
| 2010's | 2 (40.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (4)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| 1-(3-(4-chlorobenzoyl)propyl)-4-hydroxy-4-(4-chlorophenyl)piperidine | Rattus norvegicus (Norway rat) | Ki | 0.3500 | 1 | 1 |
| gw 803430 | Rattus norvegicus (Norway rat) | Ki | 0.0003 | 1 | 1 |
| t-226296 | Rattus norvegicus (Norway rat) | IC50 | 0.0240 | 1 | 1 |
| snap7941 | Rattus norvegicus (Norway rat) | Ki | 0.0008 | 3 | 3 |