Proteins > Glutamate receptor 1
Page last updated: 2024-08-07 13:07:58

Glutamate receptor 1

A glutamate receptor 1 that is encoded in the genome of mouse. [OMA:P23818, PRO:DNx]

Synonyms

GluR-1;
AMPA-selective glutamate receptor 1;
GluR-A;
GluR-K1;
Glutamate receptor ionotropic, AMPA 1;
GluA1

Research

Bioassay Publications (4)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's3 (75.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (8)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acidMus musculus (house mouse)IC500.040011
quisqualic acidMus musculus (house mouse)IC500.080011
4-bromohomoibotenic acid, (rs)-isomerMus musculus (house mouse)IC500.600011
4-bromohomoibotenic acidMus musculus (house mouse)IC5032.000011
tqx 173Mus musculus (house mouse)IC502.300011

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acidMus musculus (house mouse)EC508.700011
4-bromohomoibotenic acid, (rs)-isomerMus musculus (house mouse)EC5014.000011

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
gyki 52466Mus musculus (house mouse)ED5030.550022
cfm 2Mus musculus (house mouse)ED5013.800022
4,5-dihydro-7,8-dimethoxy-1-phenyl-3h-2,3-benzodiazepin-4-oneMus musculus (house mouse)ED5032.850022