Page last updated: 2024-08-07 13:03:25
Substance-K receptor
A substance-K receptor that is encoded in the genome of rat. [OMA:P16610, PRO:DNx]
Synonyms
SKR;
NK-2 receptor;
NK-2R;
Neurokinin A receptor;
Tachykinin receptor 2
Research
Bioassay Publications (7)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 5 (71.43) | 18.2507 |
| 2000's | 1 (14.29) | 29.6817 |
| 2010's | 1 (14.29) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (10)
Drugs with Inhibition Measurements
Drugs with Activation Measurements
Design and synthesis of side-chain conformationally restricted phenylalanines and their use for structure-activity studies on tachykinin NK-1 receptor.Journal of medicinal chemistry, , May-27, Volume: 37, Issue:11, 1994
Conformationally constrained tachykinin analogues: potent and highly selective neurokinin NK-2 receptor agonists.Journal of medicinal chemistry, , Oct-30, Volume: 35, Issue:22, 1992
Allosteric functional switch of neurokinin A-mediated signaling at the neurokinin NK2 receptor: structural exploration.Journal of medicinal chemistry, , Oct-08, Volume: 52, Issue:19, 2009
Conformationally constrained tachykinin analogues: potent and highly selective neurokinin NK-2 receptor agonists.Journal of medicinal chemistry, , Oct-30, Volume: 35, Issue:22, 1992