Page last updated: 2024-08-07 12:44:20
Sodium-dependent noradrenaline transporter
A sodium-dependent noradrenaline transporter that is encoded in the genome of mouse. [OMA:O55192, PRO:DNx]
Synonyms
Norepinephrine transporter;
NET;
Solute carrier family 6 member 2
Research
Bioassay Publications (2)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (50.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (7)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
citalopram | Mus musculus (house mouse) | Ki | 1.0000 | 1 | 1 |
cyproheptadine | Mus musculus (house mouse) | Ki | 0.2900 | 1 | 1 |
fluoxetine | Mus musculus (house mouse) | Ki | 0.0850 | 1 | 1 |
imipramine | Mus musculus (house mouse) | Ki | 0.0140 | 2 | 2 |
paroxetine | Mus musculus (house mouse) | Ki | 0.0200 | 1 | 1 |
femoxetine | Mus musculus (house mouse) | Ki | 0.1200 | 1 | 1 |
9-(aminomethyl)-9,10-dihydroanthracene | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |