Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
ipriflavone | Homo sapiens (human) | IC50 | 94.8000 | 1 | 0 |
methyldimethylaminoazobenzene | Homo sapiens (human) | IC50 | 3.7400 | 1 | 0 |
1-amino-2-methylanthraquinone | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
glaucine | Homo sapiens (human) | IC50 | 5.2350 | 2 | 0 |
Berberine chloride (TN) | Homo sapiens (human) | IC50 | 53.8300 | 2 | 0 |
2-hydroxybenzothiazole | Homo sapiens (human) | IC50 | 100.0000 | 2 | 0 |
alosetron hydrochloride | Homo sapiens (human) | IC50 | 12.6500 | 2 | 0 |
witisol | Homo sapiens (human) | IC50 | 39.3000 | 1 | 0 |
papaveraldine | Homo sapiens (human) | IC50 | 3.7350 | 2 | 0 |
12-phenyllauric acid | Homo sapiens (human) | IC50 | 100.0000 | 2 | 0 |
4',6-dihydroxyflavone | Homo sapiens (human) | IC50 | 11.6000 | 1 | 0 |
N-[2-(1-azepanyl)-1,3-benzothiazol-6-yl]carbamic acid ethyl ester | Homo sapiens (human) | IC50 | 9.4450 | 1 | 0 |
1,3(2h,4h)-isoquinolinedione | Homo sapiens (human) | IC50 | 0.3714 | 2 | 0 |
6-bromoindirubin-3'-oxime | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
trimethylcolchicinic acid | Homo sapiens (human) | IC50 | 62.8500 | 2 | 0 |
2-[(4-nitrophenyl)methylthio]-1,3-benzoxazole | Homo sapiens (human) | IC50 | 16.2000 | 1 | 0 |
N-(1,3-benzothiazol-2-yl)-N-methylbenzamide | Homo sapiens (human) | IC50 | 50.4000 | 1 | 0 |
N5,N5-dimethyl-2,1,3-benzoxadiazole-4,5-diamine | Homo sapiens (human) | IC50 | 30.1500 | 2 | 0 |
N-(2-fluorophenyl)-4-phenylmethoxybenzamide | Homo sapiens (human) | IC50 | 99.0000 | 1 | 0 |
5-amino-3-(4-methoxyphenyl)-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid ethyl ester | Homo sapiens (human) | IC50 | 6.3100 | 2 | 0 |
vu0038882 | Homo sapiens (human) | IC50 | 19.3000 | 1 | 0 |
2-[(2-fluorophenyl)methylthio]-5-(4-methylphenyl)-1,3,4-oxadiazole | Homo sapiens (human) | IC50 | 21.4000 | 1 | 0 |
[4-[(2-fluorophenyl)methoxy]phenyl]-(1-pyrrolidinyl)methanethione | Homo sapiens (human) | IC50 | 2.3800 | 2 | 0 |
4-methyl-N,5-diphenyl-3-thiophenecarboxamide | Homo sapiens (human) | IC50 | 7.4700 | 1 | 0 |
js 3 | Homo sapiens (human) | IC50 | 29.8000 | 1 | 0 |
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-4-methylbenzamide | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
5-amino-3-(2-methylphenyl)-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid ethyl ester | Homo sapiens (human) | IC50 | 10.7100 | 2 | 0 |
2-[[anilino(oxo)methyl]amino]-N-(phenylmethyl)benzamide | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
5-[(4-methylphenoxy)methyl]-3-phenyl-1,2,4-oxadiazole | Homo sapiens (human) | IC50 | 69.9000 | 1 | 0 |
3-amino-2-(4-methylphenyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
N-(3-methoxyphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide | Homo sapiens (human) | IC50 | 18.9000 | 1 | 0 |
N-(1-naphthalenyl)-5-pyridin-4-yl-1,3,4-thiadiazol-2-amine | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
2',4',6'-Trihydroxydihydrochalcone | Homo sapiens (human) | IC50 | 100.0000 | 2 | 0 |
2-(4-hydroxyphenyl)-5-methyl-1H-pyrazol-3-one | Homo sapiens (human) | IC50 | 18.1500 | 2 | 0 |
5-(2-chlorophenyl)-N-phenyl-2-furancarboxamide | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
N-(4-methylphenyl)-4-benzofuro[3,2-d]pyrimidinamine | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
4-(2-quinoxalinylamino)benzoic acid ethyl ester | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
4-(3-chloro-2-thiophenyl)-2-(3-pyridinyl)thiazole | Homo sapiens (human) | IC50 | 22.6000 | 1 | 0 |
2-chloro-3-(prop-2-enylamino)naphthalene-1,4-dione | Homo sapiens (human) | IC50 | 10.1000 | 1 | 0 |
fm19g11 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
5-bromo-N-(4,7-dimethoxy-1,3-benzothiazol-2-yl)-2-thiophenecarboxamide | Homo sapiens (human) | IC50 | 99.0000 | 1 | 0 |
3-[[[3-[(3-nitrophenyl)sulfamoyl]phenyl]-oxomethyl]amino]benzoic acid | Homo sapiens (human) | IC50 | 11.9000 | 1 | 0 |
2,4-dithiophen-2-ylthiazole | Homo sapiens (human) | IC50 | 28.2000 | 1 | 0 |
4-(4-methylphenyl)-2-(3-nitrophenyl)-3-pyrazolamine | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
4b,9b-dihydroxy-7,8-dihydro-6H-indeno[1,2-b]benzofuran-9,10-dione | Homo sapiens (human) | IC50 | 4.5850 | 2 | 0 |
4-methylbenzenesulfonic acid [4-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-methoxyphenyl] ester | Homo sapiens (human) | IC50 | 27.9000 | 2 | 0 |
benzenesulfonic acid [4-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-methoxyphenyl] ester | Homo sapiens (human) | IC50 | 59.0500 | 2 | 0 |
4-[[1-[(3,4-dichlorophenyl)methyl]-3-indolyl]-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-one | Homo sapiens (human) | IC50 | 6.0000 | 2 | 0 |
benzenesulfonic acid [4-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-ethoxyphenyl] ester | Homo sapiens (human) | IC50 | 27.0500 | 2 | 0 |
N-[(2-chlorophenyl)methyl]-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-hydroxy-5-nitro-4-triazolimine | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
3,4-dihydro-1H-isoquinolin-2-yl-(1-ethylsulfonyl-4-piperidinyl)methanone | Homo sapiens (human) | IC50 | 54.4450 | 2 | 0 |
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-(1-phenylethylamino)ethyl] ester | Homo sapiens (human) | IC50 | 11.8250 | 2 | 0 |
4-[(4-ethoxy-3-methoxyphenyl)-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-one | Homo sapiens (human) | IC50 | 38.2500 | 2 | 0 |
5-methyl-4-[(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)-[1-(1-naphthalenylmethyl)-3-indolyl]methyl]-1,2-dihydropyrazol-3-one | Homo sapiens (human) | IC50 | 4.3400 | 2 | 0 |
5-(2-chlorophenyl)-N-(4-methoxyphenyl)-2-furancarboxamide | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-[(phenylmethyl)amino]ethyl] ester | Homo sapiens (human) | IC50 | 12.9000 | 1 | 0 |
2-[4-(difluoromethylthio)anilino]benzoic acid [2-(dimethylamino)-2-oxoethyl] ester | Homo sapiens (human) | IC50 | 17.8000 | 1 | 0 |
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-[[oxo-[(phenylmethyl)amino]methyl]amino]ethyl] ester | Homo sapiens (human) | IC50 | 4.2800 | 1 | 0 |
2'-hydroxy-4-methoxychalcone | Homo sapiens (human) | IC50 | 10.6000 | 1 | 0 |
reumycin | Homo sapiens (human) | IC50 | 1.8500 | 2 | 0 |
nifuratrone | Homo sapiens (human) | IC50 | 30.0500 | 2 | 0 |
(5-ethyl-8-methyl-[1,2,4]triazino[5,6-b]indol-3-yl)hydrazine | Homo sapiens (human) | IC50 | 54.4200 | 2 | 0 |
5-chloro-N-[4-(2-thiazolo[5,4-b]pyridinyl)phenyl]-2-thiophenesulfonamide | Homo sapiens (human) | IC50 | 29.1000 | 1 | 0 |
dihydroxanthohumol | Homo sapiens (human) | IC50 | 13.3000 | 1 | 0 |
3-[3,5-dimethyl-1-[6-(1-piperidinyl)-3-pyridazinyl]-4-pyrazolyl]-N-(3-fluoro-4-methylphenyl)propanamide | Homo sapiens (human) | IC50 | 29.4000 | 1 | 0 |
2-chloro-3-[2-(4-methylphenyl)-5-tetrazolyl]pyridine | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
(2S)-2-[[[1-[(2S)-3-methyl-2-[(4-methylphenyl)sulfonylamino]-1-oxobutyl]-4-piperidinyl]-oxomethyl]amino]-2-phenylacetic acid | Homo sapiens (human) | IC50 | 100.0000 | 2 | 0 |
3-chloro-N-propan-2-yl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamide | Homo sapiens (human) | IC50 | 69.3000 | 1 | 0 |
1-(2,3-dihydro-1H-inden-5-yl)-3-(2-ethoxyphenyl)urea | Homo sapiens (human) | IC50 | 9.2900 | 1 | 0 |
2-(4-methoxyphenyl)-1H-quinazolin-4-one | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |