Page last updated: 2024-08-07 12:35:10

vasopressin V1b receptor

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (32)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
9-xylosyladenineHomo sapiens (human)Potency9.765410
pentoxifyllineHomo sapiens (human)Potency38.876910
2-chloroadenosineHomo sapiens (human)Potency19.438410
phenylisopropyladenosineHomo sapiens (human)Potency21.862110
n(6)-phenyladenosineHomo sapiens (human)Potency30.881010
n-methyladenosineHomo sapiens (human)Potency61.615710
adenosine amine congenerHomo sapiens (human)Potency2.745810
adenosine-5'-(n-ethylcarboxamide)Homo sapiens (human)Potency1.943810
n(6)-cyclopentyladenosineHomo sapiens (human)Potency30.881010
1-[1-(4-methoxyphenyl)-4-pyrazolo[3,4-d]pyrimidinyl]-4-piperidinecarboxamideHomo sapiens (human)Potency24.529710
5-(5-chloro-2-methoxyphenyl)-3H-1,3,4-oxadiazole-2-thioneHomo sapiens (human)Potency4.351710
N-(5-acetyl-4-methyl-2-thiazolyl)-2-methylpropanamideHomo sapiens (human)Potency17.324510
8-methyl-1,5-dihydropyrimido[5,4-b]indole-4-thioneHomo sapiens (human)Potency6.147010
3-[[[5-(phenylmethyl)-1,3,4-oxadiazol-2-yl]thio]methyl]benzoic acidHomo sapiens (human)Potency27.457510
5-chloro-N-(2-furanylmethyl)-2-[[(4-methoxyphenyl)-oxomethyl]amino]benzamideHomo sapiens (human)Potency59.508110
2-[[3-cyano-6-(4-methylphenyl)-4-(trifluoromethyl)-2-pyridinyl]thio]-N-(4-methoxyphenyl)acetamideHomo sapiens (human)Potency17.324510
4-(1,3-dioxo-2-isoindolyl)-N-(4-methyl-2-pyrimidinyl)benzenesulfonamideHomo sapiens (human)Potency14.947810
N-(2-ethylphenyl)-2-[[2-(4-methoxyphenyl)-4-oxo-1-benzopyran-6-yl]oxy]acetamideHomo sapiens (human)Potency19.438410
LSM-28559Homo sapiens (human)Potency43.620610
8-chloro-N-(4-fluorophenyl)-2-(2-pyridinyl)-4-quinolinecarboxamideHomo sapiens (human)Potency17.324510
6-(4-bromophenyl)-3-methyl-1-[2-(2H-tetrazol-5-yl)ethyl]-4-(trifluoromethyl)pyrazolo[3,4-b]pyridineHomo sapiens (human)Potency17.324510
4-amino-7,8,9,10-tetrahydro-6H-pyrimido[3,4]pyrrolo[3,5-a]azepine-11-carbonitrileHomo sapiens (human)Potency34.649110
1-cyclopentyl-2-imino-10-methyl-5-oxo-N-(2-oxolanylmethyl)-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxamideHomo sapiens (human)Potency38.876910
2-[[2-(1-adamantyl)-2-oxoethyl]thio]-6-amino-4-(4-chlorophenyl)pyridine-3,5-dicarbonitrileHomo sapiens (human)Potency12.264810
N-(1,3-dioxo-5-isoindolyl)-1,3-benzothiazole-6-carboxamideHomo sapiens (human)Potency21.810310
2-(1,3-dimethyl-2,6-dioxo-7-purinyl)-N'-[2-(2-ethoxyphenoxy)-1-oxoethyl]acetohydrazideHomo sapiens (human)Potency30.881010
N-[5-(1-azepanylsulfonyl)-2-chlorophenyl]-2-[(4-methyl-1,2,4-triazol-3-yl)thio]acetamideHomo sapiens (human)Potency10.957010
sulfuretinHomo sapiens (human)Potency43.620610
8-(1-piperidinylsulfonyl)-6-pyrido[1,2-a]quinazolinoneHomo sapiens (human)Potency43.620610
1-(2-phenylethyl)-4-([1,2,4]triazolo[4,3-a]quinoxalin-4-yl)piperazine-2,6-dioneHomo sapiens (human)Potency24.471610
bucladesineHomo sapiens (human)Potency1.376110
cyclic amp, monosodium saltHomo sapiens (human)Potency0.194410