Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
2-fluoroadenosine | | Potency | 1.9857 | 1 | 0 |
triphenyltetrazolium chloride | | Potency | 24.9988 | 1 | 0 |
s-2678 | | Potency | 22.2802 | 1 | 0 |
triclabendazole | | Potency | 88.6991 | 1 | 0 |
2,2',2''-terpyridine | | Potency | 3.5312 | 1 | 0 |
cycloadiphenine hydrochloride | | Potency | 14.0579 | 1 | 0 |
sb 205384 | | Potency | 22.2802 | 1 | 0 |
anisomycin | | Potency | 7.0456 | 1 | 0 |
nsc689857 | | Potency | 3.9620 | 1 | 0 |
4-methyl-N-(pyridin-4-ylmethyl)benzenesulfonamide | | Potency | 2.2280 | 1 | 0 |
4-[1-(4-hydroxyphenyl)ethenyl]phenol | | Potency | 14.0579 | 1 | 0 |
2,6-dimethyl-4-(1-phenyl-4-pyrazolyl)furo[2,3-d]pyrimidine | | Potency | 15.7732 | 1 | 0 |
N-[7-(1-oxopropyl)-2,3-dihydro-1,4-benzodioxin-6-yl]benzamide | | Potency | 3.9620 | 1 | 0 |
4-methyl-N-(3-nitrophenyl)-5-phenyl-3-thiophenecarboxamide | | Potency | 11.1666 | 1 | 0 |
2-[[3-cyano-6-(4-methoxyphenyl)-4-phenyl-2-pyridinyl]thio]-N-(5-methyl-2-thiazolyl)acetamide | | Potency | 19.8573 | 1 | 0 |
N-[2-(trifluoromethyl)-1,3-benzodioxol-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide | | Potency | 24.9988 | 1 | 0 |
3-[5-[(4-chlorophenyl)methylthio]-1,3,4-oxadiazol-2-yl]-1-(phenylmethyl)-2-pyridinone | | Potency | 12.5291 | 1 | 0 |
N2,N2-dimethyl-6-[[[1-(1-naphthalenyl)-5-tetrazolyl]thio]methyl]-1,3,5-triazine-2,4-diamine | | Potency | 5.5965 | 1 | 0 |
4-[(2,4-dichlorophenoxy)methyl]-N-[2-(dimethylamino)ethyl]benzamide | | Potency | 15.7732 | 1 | 0 |
4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-N-[4-(1-pyrrolidinylsulfonyl)phenyl]benzamide | | Potency | 0.6279 | 1 | 0 |
1,2,3,4-tetrahydroacridine-9-carboxylic acid [2-(3-chloro-4-methoxyanilino)-2-oxoethyl] ester | | Potency | 4.9879 | 1 | 0 |
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(3,5-dimethyl-1-pyrazolyl)benzamide | | Potency | 9.9522 | 1 | 0 |
3,3-dimethyl-1-[[9-(methylthio)-5,6-dihydrothieno[3,4-h]quinazolin-2-yl]thio]-2-butanone | | Potency | 24.9988 | 1 | 0 |
N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamide | | Potency | 9.9522 | 1 | 0 |
4-[(1-methyl-2-oxo-4-quinolinyl)oxy]-N-(4-methyl-2-pyridinyl)butanamide | | Potency | 7.9053 | 1 | 0 |
N-(5-chloro-2-methoxyphenyl)-2,4-dimethyl-5-oxazolecarboxamide | | Potency | 12.5291 | 1 | 0 |
4-[2-[[2-[[4-(1,3-benzodioxol-5-yl)-2-thiazolyl]amino]-2-oxoethyl]thio]-1-oxoethyl]-1-piperazinecarboxylic acid ethyl ester | | Potency | 15.7732 | 1 | 0 |
2-[[3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-2-thieno[3,2-d]pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamide | | Potency | 11.1666 | 1 | 0 |
6-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-5-thieno[2,3-b]pyrrolecarboxylic acid methyl ester | | Potency | 7.9053 | 1 | 0 |
N-[3-(3,5-dimethyl-1-piperidinyl)propyl]-1-[[5-methyl-2-(2-methylphenyl)-4-oxazolyl]methyl]-4-piperidinecarboxamide | | Potency | 1.4058 | 1 | 0 |
2-[2-(2-chlorophenyl)-1-benzimidazolyl]-N-(2-propan-2-ylphenyl)acetamide | | Potency | 8.8699 | 1 | 0 |
nsc 105827 | | Potency | 0.4445 | 1 | 0 |
2-(N-(2-chloro-1-oxoethyl)-3-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamide | | Potency | 0.8870 | 1 | 0 |
2-ethyl-4-[[(3-methyl-2-benzofuranyl)-oxomethyl]amino]-1H-1,5-benzodiazepine-3-carboxylic acid ethyl ester | | Potency | 12.5291 | 1 | 0 |
N-[3-(1,3-dioxo-2-benzo[de]isoquinolinyl)propyl]-N-(2-methoxy-4-methylphenyl)-2-thiophenecarboxamide | | Potency | 12.5291 | 1 | 0 |
2-(1,3-benzothiazol-2-ylmethylthio)-1-butyl-5-benzimidazolesulfonamide | | Potency | 17.6978 | 1 | 0 |
N,N-diethyl-2-[[7-[(4-methoxyphenyl)methyl]-8-oxo-[1,3]dioxolo[4,5-g]quinazolin-6-yl]thio]acetamide | | Potency | 5.5965 | 1 | 0 |
3-methoxy-N-[4-methyl-2-(4-morpholinyl)-6-quinolinyl]benzamide | | Potency | 2.8049 | 1 | 0 |
7-chloro-N-(phenylmethyl)-4-quinolinamine | | Potency | 9.9522 | 1 | 0 |
4-hydroxyestradiol | | Potency | 19.8573 | 1 | 0 |
4-amino-5-chloro-N-[(3R,4S)-1-[3-(4-fluorophenoxy)propyl]-3-methoxy-4-piperidinyl]-2-methoxybenzamide | | Potency | 4.4455 | 1 | 0 |
arteannuin b | | Potency | 31.4716 | 1 | 0 |
2-(2,4-dimethoxyphenyl)-5-methyl-4-[[4-(4-quinazolinyl)-1-piperazinyl]methyl]oxazole | | Potency | 4.9879 | 1 | 0 |
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-4-methyl-5-thiadiazolecarboxamide | | Potency | 3.1472 | 1 | 0 |
4-[4-[(1-methyl-5-tetrazolyl)thio]-5-thieno[2,3-d]pyrimidinyl]benzonitrile | | Potency | 24.9988 | 1 | 0 |