Page last updated: 2024-08-07 15:10:09

alternatively spliced Trp4

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (60)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
ml 204Mus musculus (house mouse)IC501.690050

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
methylbufoteninMus musculus (house mouse)EC500.670010
2,5-di-tert-butylhydroquinoneMus musculus (house mouse)EC500.376010
fluspirileneMus musculus (house mouse)EC506.682710
spiperoneMus musculus (house mouse)EC506.682710
acetylcholine chlorideMus musculus (house mouse)EC500.421310
diphenylguanidineMus musculus (house mouse)EC5010.590710
c 137Mus musculus (house mouse)EC501.333310
acetylcholine bromideMus musculus (house mouse)EC500.066710
oxymetazoline hydrochlorideMus musculus (house mouse)EC503.350010
1-(10-methyl-2-phenothiazinyl)ethanoneMus musculus (house mouse)EC507.497310
ml 204Mus musculus (house mouse)EC500.002710
2-[(6-butoxy-3-pyridinyl)amino]-4-chlorobenzoic acidMus musculus (house mouse)EC5010.590710
chondocurine (1beta)-(+-)-isomerMus musculus (house mouse)EC501.333310
N-butyl-1H-benzimidazol-2-amineMus musculus (house mouse)EC502.985310
ua8967Mus musculus (house mouse)EC505.956010
3-[[cyclopentyl-[[1-(phenylmethyl)-5-tetrazolyl]methyl]amino]methyl]-8-methyl-1H-quinolin-2-oneMus musculus (house mouse)EC500.149310
5-ethyl-3-[(2-fluorophenyl)methyl]-N-[2-(2-pyridinyl)ethyl]-7-triazolo[4,5-d]pyrimidinamineMus musculus (house mouse)EC502.660010
1-[5-(2-amino-5-methyl-4-thiazolyl)-2,3-dihydroindol-1-yl]-1-butanoneMus musculus (house mouse)EC500.376010
methamilane methiodideMus musculus (house mouse)EC500.188010
4-[1-(4-hydroxyphenyl)ethenyl]phenolMus musculus (house mouse)EC503.757310
2-ethyl-1-[(2-methoxyphenyl)methyl]benzimidazoleMus musculus (house mouse)EC5010.590710
N-(4,6-dimethyl-2-pyrimidinyl)-1,3-bis(phenylmethyl)-2,4-dihydro-1,3,5-triazin-6-amineMus musculus (house mouse)EC504.730710
4-(1-benzotriazolyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidineMus musculus (house mouse)EC506.682710
2,6-dimethyl-N-(4-methylphenyl)-4-quinolinamineMus musculus (house mouse)EC501.496010
N-[3-(methylthio)-1,2,4-thiadiazol-5-yl]-2-phenylacetamideMus musculus (house mouse)EC505.308010
4-[[[[oxo-(4-phenylphenyl)methyl]amino]-sulfanylidenemethyl]amino]benzoic acidMus musculus (house mouse)EC504.730710
5-bromo-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamideMus musculus (house mouse)EC500.841310
N-[[3-(4-fluorophenyl)-1-phenyl-4-pyrazolyl]methyl]-1-phenylmethanamineMus musculus (house mouse)EC505.308010
5-(4-chlorophenyl)-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamideMus musculus (house mouse)EC500.066710
4-methyl-N-[(1-oxopentylhydrazo)-sulfanylidenemethyl]benzamideMus musculus (house mouse)EC502.985310
5-bromo-N-[[[oxo(thiophen-2-yl)methyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)EC505.308010
N-[[[(2-methylphenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]benzamideMus musculus (house mouse)EC502.113310
4,5-dichloro-2-methyl-1-(2-phenoxyethyl)imidazoleMus musculus (house mouse)EC505.308010
5,6-dimethyl-N-[2-methyl-2-(4-morpholinyl)propyl]-4-thieno[2,3-d]pyrimidinamineMus musculus (house mouse)EC500.841310
1-(2-chlorophenoxy)-3-(2-methyl-1-benzimidazolyl)-2-propanolMus musculus (house mouse)EC503.349310
2,2'-[3-(2-methoxyphenyl)-1,2-propanediyl]bis(1H-benzimidazole)Mus musculus (house mouse)EC503.349310
2-[[(4-chlorophenyl)thio]methyl]-5-methylimidazo[1,2-a]pyridineMus musculus (house mouse)EC504.216010
4-chloro-N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideMus musculus (house mouse)EC501.058710
N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideMus musculus (house mouse)EC500.749310
N-[3-(3,5-dimethyl-1-piperidinyl)propyl]-2-[(1-methyl-2-oxo-4-quinolinyl)oxy]acetamideMus musculus (house mouse)EC500.749310
N-(2-furanylmethyl)-5,7-dimethyl-6-[(3-methylphenyl)methyl]-3-pyrazolo[1,5-a]pyrimidinecarboxamideMus musculus (house mouse)EC503.760010
2-[(2,2-dimethyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)oxy]-N-heptylacetamideMus musculus (house mouse)EC500.944010
N-(3-chlorophenyl)-5-oxo-9b-phenyl-2,3-dihydroimidazo[2,1-a]isoindole-1-carboxamideMus musculus (house mouse)EC503.757310
N-(4-phenylmethoxyphenyl)-3-[4-(phenylmethyl)-1-piperazinyl]propanamideMus musculus (house mouse)EC500.130010
2-(1H-indol-3-yl)-8-methylimidazo[1,2-a]pyridineMus musculus (house mouse)EC505.956010
2-[4-[[[[(2,4-dichlorophenyl)-oxomethyl]amino]-sulfanylidenemethyl]amino]-3-methylphenyl]-3,3,3-trifluoro-2-hydroxypropanoic acid ethyl esterMus musculus (house mouse)EC503.350010
1-(3-chlorophenyl)-3-[2-(dimethylamino)-2-phenylethyl]thioureaMus musculus (house mouse)EC500.596010
1-[3-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-4-methoxyphenyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acidMus musculus (house mouse)EC500.530710
2-thiophen-2-yl-N-(thiophen-2-ylmethyl)-4-quinazolinamineMus musculus (house mouse)EC504.730710
1-Ethyl-9H-pyrido[3,4-b]indoleMus musculus (house mouse)EC502.985310
dihydrothobainoneMus musculus (house mouse)EC500.042710
1-(3,4-dimethylphenyl)-4-(4-methyl-1-piperidinyl)phthalazineMus musculus (house mouse)EC503.350010
lasalocid sodiumMus musculus (house mouse)EC505.956010
3,4,5-trimethoxy-N-[[[oxo-[(1S,2S)-2-phenylcyclopropyl]methyl]hydrazo]-sulfanylidenemethyl]benzamideMus musculus (house mouse)EC503.757310
(2R,4R)-4-(1-acetyl-3-indolyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-N-(phenylmethyl)-3,4-dihydro-2H-pyran-6-carboxamideMus musculus (house mouse)EC508.413310
4-methyl-N-[[(5-methyl-2,1,3-benzothiadiazol-4-yl)amino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)EC505.956010
(3-propan-2-yloxyphenyl)-[1-[(1-propan-2-yl-4-pyrazolyl)methyl]-3-piperidinyl]methanoneMus musculus (house mouse)EC502.113310
[1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(2-phenylethyl)-4-piperidinyl]methanolMus musculus (house mouse)EC508.413310
cym51010Mus musculus (house mouse)EC500.026710
N-[4-(1H-benzimidazol-2-yl)phenyl]-1-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-piperidinecarboxamideMus musculus (house mouse)EC500.000310