Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
methylbufotenin | Mus musculus (house mouse) | EC50 | 0.6700 | 1 | 0 |
2,5-di-tert-butylhydroquinone | Mus musculus (house mouse) | EC50 | 0.3760 | 1 | 0 |
fluspirilene | Mus musculus (house mouse) | EC50 | 6.6827 | 1 | 0 |
spiperone | Mus musculus (house mouse) | EC50 | 6.6827 | 1 | 0 |
acetylcholine chloride | Mus musculus (house mouse) | EC50 | 0.4213 | 1 | 0 |
diphenylguanidine | Mus musculus (house mouse) | EC50 | 10.5907 | 1 | 0 |
c 137 | Mus musculus (house mouse) | EC50 | 1.3333 | 1 | 0 |
acetylcholine bromide | Mus musculus (house mouse) | EC50 | 0.0667 | 1 | 0 |
oxymetazoline hydrochloride | Mus musculus (house mouse) | EC50 | 3.3500 | 1 | 0 |
1-(10-methyl-2-phenothiazinyl)ethanone | Mus musculus (house mouse) | EC50 | 7.4973 | 1 | 0 |
ml 204 | Mus musculus (house mouse) | EC50 | 0.0027 | 1 | 0 |
2-[(6-butoxy-3-pyridinyl)amino]-4-chlorobenzoic acid | Mus musculus (house mouse) | EC50 | 10.5907 | 1 | 0 |
chondocurine (1beta)-(+-)-isomer | Mus musculus (house mouse) | EC50 | 1.3333 | 1 | 0 |
N-butyl-1H-benzimidazol-2-amine | Mus musculus (house mouse) | EC50 | 2.9853 | 1 | 0 |
ua8967 | Mus musculus (house mouse) | EC50 | 5.9560 | 1 | 0 |
3-[[cyclopentyl-[[1-(phenylmethyl)-5-tetrazolyl]methyl]amino]methyl]-8-methyl-1H-quinolin-2-one | Mus musculus (house mouse) | EC50 | 0.1493 | 1 | 0 |
5-ethyl-3-[(2-fluorophenyl)methyl]-N-[2-(2-pyridinyl)ethyl]-7-triazolo[4,5-d]pyrimidinamine | Mus musculus (house mouse) | EC50 | 2.6600 | 1 | 0 |
1-[5-(2-amino-5-methyl-4-thiazolyl)-2,3-dihydroindol-1-yl]-1-butanone | Mus musculus (house mouse) | EC50 | 0.3760 | 1 | 0 |
methamilane methiodide | Mus musculus (house mouse) | EC50 | 0.1880 | 1 | 0 |
4-[1-(4-hydroxyphenyl)ethenyl]phenol | Mus musculus (house mouse) | EC50 | 3.7573 | 1 | 0 |
2-ethyl-1-[(2-methoxyphenyl)methyl]benzimidazole | Mus musculus (house mouse) | EC50 | 10.5907 | 1 | 0 |
N-(4,6-dimethyl-2-pyrimidinyl)-1,3-bis(phenylmethyl)-2,4-dihydro-1,3,5-triazin-6-amine | Mus musculus (house mouse) | EC50 | 4.7307 | 1 | 0 |
4-(1-benzotriazolyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine | Mus musculus (house mouse) | EC50 | 6.6827 | 1 | 0 |
2,6-dimethyl-N-(4-methylphenyl)-4-quinolinamine | Mus musculus (house mouse) | EC50 | 1.4960 | 1 | 0 |
N-[3-(methylthio)-1,2,4-thiadiazol-5-yl]-2-phenylacetamide | Mus musculus (house mouse) | EC50 | 5.3080 | 1 | 0 |
4-[[[[oxo-(4-phenylphenyl)methyl]amino]-sulfanylidenemethyl]amino]benzoic acid | Mus musculus (house mouse) | EC50 | 4.7307 | 1 | 0 |
5-bromo-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamide | Mus musculus (house mouse) | EC50 | 0.8413 | 1 | 0 |
N-[[3-(4-fluorophenyl)-1-phenyl-4-pyrazolyl]methyl]-1-phenylmethanamine | Mus musculus (house mouse) | EC50 | 5.3080 | 1 | 0 |
5-(4-chlorophenyl)-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamide | Mus musculus (house mouse) | EC50 | 0.0667 | 1 | 0 |
4-methyl-N-[(1-oxopentylhydrazo)-sulfanylidenemethyl]benzamide | Mus musculus (house mouse) | EC50 | 2.9853 | 1 | 0 |
5-bromo-N-[[[oxo(thiophen-2-yl)methyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamide | Mus musculus (house mouse) | EC50 | 5.3080 | 1 | 0 |
N-[[[(2-methylphenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]benzamide | Mus musculus (house mouse) | EC50 | 2.1133 | 1 | 0 |
4,5-dichloro-2-methyl-1-(2-phenoxyethyl)imidazole | Mus musculus (house mouse) | EC50 | 5.3080 | 1 | 0 |
5,6-dimethyl-N-[2-methyl-2-(4-morpholinyl)propyl]-4-thieno[2,3-d]pyrimidinamine | Mus musculus (house mouse) | EC50 | 0.8413 | 1 | 0 |
1-(2-chlorophenoxy)-3-(2-methyl-1-benzimidazolyl)-2-propanol | Mus musculus (house mouse) | EC50 | 3.3493 | 1 | 0 |
2,2'-[3-(2-methoxyphenyl)-1,2-propanediyl]bis(1H-benzimidazole) | Mus musculus (house mouse) | EC50 | 3.3493 | 1 | 0 |
2-[[(4-chlorophenyl)thio]methyl]-5-methylimidazo[1,2-a]pyridine | Mus musculus (house mouse) | EC50 | 4.2160 | 1 | 0 |
4-chloro-N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamide | Mus musculus (house mouse) | EC50 | 1.0587 | 1 | 0 |
N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamide | Mus musculus (house mouse) | EC50 | 0.7493 | 1 | 0 |
N-[3-(3,5-dimethyl-1-piperidinyl)propyl]-2-[(1-methyl-2-oxo-4-quinolinyl)oxy]acetamide | Mus musculus (house mouse) | EC50 | 0.7493 | 1 | 0 |
N-(2-furanylmethyl)-5,7-dimethyl-6-[(3-methylphenyl)methyl]-3-pyrazolo[1,5-a]pyrimidinecarboxamide | Mus musculus (house mouse) | EC50 | 3.7600 | 1 | 0 |
2-[(2,2-dimethyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)oxy]-N-heptylacetamide | Mus musculus (house mouse) | EC50 | 0.9440 | 1 | 0 |
N-(3-chlorophenyl)-5-oxo-9b-phenyl-2,3-dihydroimidazo[2,1-a]isoindole-1-carboxamide | Mus musculus (house mouse) | EC50 | 3.7573 | 1 | 0 |
N-(4-phenylmethoxyphenyl)-3-[4-(phenylmethyl)-1-piperazinyl]propanamide | Mus musculus (house mouse) | EC50 | 0.1300 | 1 | 0 |
2-(1H-indol-3-yl)-8-methylimidazo[1,2-a]pyridine | Mus musculus (house mouse) | EC50 | 5.9560 | 1 | 0 |
2-[4-[[[[(2,4-dichlorophenyl)-oxomethyl]amino]-sulfanylidenemethyl]amino]-3-methylphenyl]-3,3,3-trifluoro-2-hydroxypropanoic acid ethyl ester | Mus musculus (house mouse) | EC50 | 3.3500 | 1 | 0 |
1-(3-chlorophenyl)-3-[2-(dimethylamino)-2-phenylethyl]thiourea | Mus musculus (house mouse) | EC50 | 0.5960 | 1 | 0 |
1-[3-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-4-methoxyphenyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid | Mus musculus (house mouse) | EC50 | 0.5307 | 1 | 0 |
2-thiophen-2-yl-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Mus musculus (house mouse) | EC50 | 4.7307 | 1 | 0 |
1-Ethyl-9H-pyrido[3,4-b]indole | Mus musculus (house mouse) | EC50 | 2.9853 | 1 | 0 |
dihydrothobainone | Mus musculus (house mouse) | EC50 | 0.0427 | 1 | 0 |
1-(3,4-dimethylphenyl)-4-(4-methyl-1-piperidinyl)phthalazine | Mus musculus (house mouse) | EC50 | 3.3500 | 1 | 0 |
lasalocid sodium | Mus musculus (house mouse) | EC50 | 5.9560 | 1 | 0 |
3,4,5-trimethoxy-N-[[[oxo-[(1S,2S)-2-phenylcyclopropyl]methyl]hydrazo]-sulfanylidenemethyl]benzamide | Mus musculus (house mouse) | EC50 | 3.7573 | 1 | 0 |
(2R,4R)-4-(1-acetyl-3-indolyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-N-(phenylmethyl)-3,4-dihydro-2H-pyran-6-carboxamide | Mus musculus (house mouse) | EC50 | 8.4133 | 1 | 0 |
4-methyl-N-[[(5-methyl-2,1,3-benzothiadiazol-4-yl)amino]-sulfanylidenemethyl]benzamide | Mus musculus (house mouse) | EC50 | 5.9560 | 1 | 0 |
(3-propan-2-yloxyphenyl)-[1-[(1-propan-2-yl-4-pyrazolyl)methyl]-3-piperidinyl]methanone | Mus musculus (house mouse) | EC50 | 2.1133 | 1 | 0 |
[1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(2-phenylethyl)-4-piperidinyl]methanol | Mus musculus (house mouse) | EC50 | 8.4133 | 1 | 0 |
cym51010 | Mus musculus (house mouse) | EC50 | 0.0267 | 1 | 0 |
N-[4-(1H-benzimidazol-2-yl)phenyl]-1-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-piperidinecarboxamide | Mus musculus (house mouse) | EC50 | 0.0003 | 1 | 0 |