Page last updated: 2024-09-03

ym 12617 and yohimbine

ym 12617 has been researched along with yohimbine in 2 studies

Compound Research Comparison

Studies
(ym 12617)
Trials
(ym 12617)
Recent Studies (post-2010)
(ym 12617)
Studies
(yohimbine)
Trials
(yohimbine)
Recent Studies (post-2010) (yohimbine)
32265,893253532

Protein Interaction Comparison

ProteinTaxonomyym 12617 (IC50)yohimbine (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.0353
Cytochrome P450 2D6Homo sapiens (human)1.02
D(2) dopamine receptorHomo sapiens (human)2.06
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)1.3
Alpha-2B adrenergic receptorHomo sapiens (human)0.0428
Alpha-2C adrenergic receptorHomo sapiens (human)0.0466
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.126
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)1.3
Alpha-1D adrenergic receptorHomo sapiens (human)1.013
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.126
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.074
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)1.3
5-hydroxytryptamine receptor 6Homo sapiens (human)1.689

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19901 (50.00)18.7374
1990's1 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Daly, CJ; Dunn, WR; McGrath, JC; Wilson, VG1
Blaylock, NA; Wilson, VG1

Other Studies

2 other study(ies) available for ym 12617 and yohimbine

ArticleYear
An attempt at selective protection from phenoxybenzamine of postjunctional alpha-adrenoceptor subtypes mediating contractions to noradrenaline in the rabbit isolated saphenous vein.
    British journal of pharmacology, 1988, Volume: 95, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Saphenous Vein; Sulfonamides; Yohimbine

1988
Pharmacological characterization of noradrenaline-induced contractions of the porcine isolated palmar lateral vein and palmar common digital artery.
    British journal of pharmacology, 1995, Volume: 114, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Arteries; Berberine; Drug Interactions; Drug Synergism; Forelimb; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Prazosin; Receptors, Adrenergic, alpha; Reproducibility of Results; Sulfonamides; Swine; Veins; Yohimbine

1995