Page last updated: 2024-09-05

rs 127445 and yohimbine

rs 127445 has been researched along with yohimbine in 1 studies

Compound Research Comparison

Studies
(rs 127445)
Trials
(rs 127445)
Recent Studies (post-2010)
(rs 127445)
Studies
(yohimbine)
Trials
(yohimbine)
Recent Studies (post-2010) (yohimbine)
291185,893253532

Protein Interaction Comparison

ProteinTaxonomyrs 127445 (IC50)yohimbine (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.0353
Cytochrome P450 2D6Homo sapiens (human)1.02
D(2) dopamine receptorHomo sapiens (human)2.06
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)1.3
Alpha-2B adrenergic receptorHomo sapiens (human)0.0428
Alpha-2C adrenergic receptorHomo sapiens (human)0.0466
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.126
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)1.3
Alpha-1D adrenergic receptorHomo sapiens (human)1.013
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.126
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.074
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)1.3
5-hydroxytryptamine receptor 6Homo sapiens (human)1.689

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bonhaus, DW; Chang, LK; Dawson, M; Eglen, RM; Flippin, LA; Greenhouse, RJ; Jaime, S; Leung, E; Martin, GR; Pulido-Rios, T; Rocha, C; Van Natta, K; Webber, A1

Other Studies

1 other study(ies) available for rs 127445 and yohimbine

ArticleYear
RS-127445: a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist.
    British journal of pharmacology, 1999, Volume: 127, Issue:5

    Topics: Animals; Calcium; CHO Cells; Cricetinae; Humans; Male; Muscle Contraction; Pyrimidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Vasodilation

1999