Page last updated: 2024-09-05

rs 127445 and ritanserin

rs 127445 has been researched along with ritanserin in 5 studies

Compound Research Comparison

Studies
(rs 127445)
Trials
(rs 127445)
Recent Studies (post-2010)
(rs 127445)
Studies
(ritanserin)
Trials
(ritanserin)
Recent Studies (post-2010) (ritanserin)
291187357571

Protein Interaction Comparison

ProteinTaxonomyrs 127445 (IC50)ritanserin (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0012
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.001
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.047
Diacylglycerol kinase alphaHomo sapiens (human)9
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.047
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0025
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0025
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0012
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.047
D(2) dopamine receptorRattus norvegicus (Norway rat)0.012

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (20.00)18.2507
2000's1 (20.00)29.6817
2010's2 (40.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Bonhaus, DW; Chang, LK; Dawson, M; Eglen, RM; Flippin, LA; Greenhouse, RJ; Jaime, S; Leung, E; Martin, GR; Pulido-Rios, T; Rocha, C; Van Natta, K; Webber, A1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Abdel-Raziq, MS; Gabr, MT1
Chen, Z; Collier, T; Fu, H; Liang, SH; Rong, J; Zhou, J1
Hong, JH; Ikeda, M; Jeong, B; Kawaguchi, K; Kim, J; Lee, KJ; Mohammad, S; Morioka, E; Ozaki, T; Takeuchi, K1

Reviews

1 review(s) available for rs 127445 and ritanserin

ArticleYear
Positron Emission Tomography (PET) Imaging Tracers for Serotonin Receptors.
    Journal of medicinal chemistry, 2022, 08-25, Volume: 65, Issue:16

    Topics: Brain; Humans; Ligands; Positron-Emission Tomography; Radiopharmaceuticals; Receptors, Serotonin

2022

Other Studies

4 other study(ies) available for rs 127445 and ritanserin

ArticleYear
RS-127445: a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist.
    British journal of pharmacology, 1999, Volume: 127, Issue:5

    Topics: Animals; Calcium; CHO Cells; Cricetinae; Humans; Male; Muscle Contraction; Pyrimidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Vasodilation

1999
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Pharmacophore-based tailoring of biphenyl amide derivatives as selective 5-hydroxytryptamine 2B receptor antagonists.
    MedChemComm, 2018, Jun-01, Volume: 9, Issue:6

    Topics:

2018
Serotonin-2C receptor involved serotonin-induced Ca²⁺ mobilisations in neuronal progenitors and neurons in rat suprachiasmatic nucleus.
    Scientific reports, 2014, Feb-17, Volume: 4

    Topics: Action Potentials; Animals; Calcium; Cells, Cultured; In Vitro Techniques; Indoles; Male; Neurons; Patch-Clamp Techniques; Piperazines; Pyridines; Pyrimidines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Ritanserin; Serotonin; Stem Cells; Suprachiasmatic Nucleus; Transcriptome

2014