Page last updated: 2024-09-02

r 56865 and glyburide

r 56865 has been researched along with glyburide in 4 studies

Compound Research Comparison

Studies
(r 56865)
Trials
(r 56865)
Recent Studies (post-2010)
(r 56865)
Studies
(glyburide)
Trials
(glyburide)
Recent Studies (post-2010) (glyburide)
72106,5546201,344

Protein Interaction Comparison

ProteinTaxonomyr 56865 (IC50)glyburide (IC50)
ATP-binding cassette sub-family C member 9Homo sapiens (human)0.22
Bile salt export pumpRattus norvegicus (Norway rat)5.7
Bile salt export pumpHomo sapiens (human)5.5333
Cytochrome P450 2C9 Homo sapiens (human)1.602
ATP-binding cassette sub-family C member 8Homo sapiens (human)0.0043
ATP-sensitive inward rectifier potassium channel 11Homo sapiens (human)0.1121
NACHT, LRR and PYD domains-containing protein 3 Mus musculus (house mouse)10
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)1.8

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gwilt, M; Henderson, CG; Orme, J; Rourke, JD1
Hoff, P; Tegtmeier, F; Xie, Y; Zacharias, E1
Lawrence, C; Rodrigo, GC1
Arita, M; Li, Y; Sato, T1

Other Studies

4 other study(ies) available for r 56865 and glyburide

ArticleYear
Effects of drugs on ventricular fibrillation and ischaemic K+ loss in a model of ischaemia in perfused guinea-pig hearts in vitro.
    European journal of pharmacology, 1992, Sep-22, Volume: 220, Issue:2-3

    Topics: 4-Aminopyridine; Animals; Anti-Arrhythmia Agents; Benzothiazoles; Calcium Channel Blockers; Disease Models, Animal; Glipizide; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Myocardial Ischemia; Piperidines; Potassium; Potassium Channels; Pyrazines; Pyridines; Sympatholytics; Thiazoles; Ventricular Fibrillation

1992
Ion channel involvement in anoxic depolarization induced by cardiac arrest in rat brain.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1995, Volume: 15, Issue:4

    Topics: Adenosine Triphosphate; Animals; Benzothiazoles; Calcium; Dizocilpine Maleate; Flunarizine; Glyburide; Heart Arrest; Hypoxia; Ion Channels; Male; Nimodipine; Piperidines; Potassium; Potassium Channels; Quinoxalines; Rats; Rats, Wistar; Sodium; Thiazoles

1995
A Na+-activated K+ current (IK,Na) is present in guinea-pig but not rat ventricular myocytes.
    Pflugers Archiv : European journal of physiology, 1999, Volume: 437, Issue:6

    Topics: Animals; Benzothiazoles; Calcium; Calcium Channel Blockers; Diltiazem; Electric Conductivity; Glyburide; Guinea Pigs; Heart; Magnesium; Male; Membrane Potentials; Patch-Clamp Techniques; Piperidines; Potassium; Potassium Channels; Rats; Rats, Sprague-Dawley; Sodium; Sodium-Potassium-Exchanging ATPase; Thiazoles; Ventricular Function

1999
Bepridil blunts the shortening of action potential duration caused by metabolic inhibition via blockade of ATP-sensitive K(+) channels and Na(+)-activated K(+) channels.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:2

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Anti-Arrhythmia Agents; Benzothiazoles; Bepridil; Calcium Channel Blockers; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Dose-Response Relationship, Drug; Glyburide; Guinea Pigs; Heart Ventricles; In Vitro Techniques; Patch-Clamp Techniques; Perfusion; Piperidines; Potassium Channels; Sodium; Thiazoles; Time Factors; Uncoupling Agents

1999