Page last updated: 2024-09-02

npc 12626 and diazepam

npc 12626 has been researched along with diazepam in 6 studies

Compound Research Comparison

Studies
(npc 12626)
Trials
(npc 12626)
Recent Studies (post-2010)
(npc 12626)
Studies
(diazepam)
Trials
(diazepam)
Recent Studies (post-2010) (diazepam)
550018,3772,3291,790

Protein Interaction Comparison

ProteinTaxonomynpc 12626 (IC50)diazepam (IC50)
Gamma-aminobutyric acid receptor subunit piHomo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit deltaHomo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit alpha-1Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit beta-1Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit alpha-2Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit alpha-3Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit beta-1Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit gamma-2Homo sapiens (human)0.0124
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0108
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0227
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit alpha-4Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit gamma-2Bos taurus (cattle)0.0266
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0106
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit beta-3Homo sapiens (human)0.0124
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit alpha-5Homo sapiens (human)0.0124
Gamma-aminobutyric acid receptor subunit alpha-3Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit alpha-2Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit beta-2Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit alpha-4Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit epsilonHomo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit alpha-6Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit gamma-1Homo sapiens (human)0.0101
GABA theta subunitRattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit gamma-3Homo sapiens (human)0.0101
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0108
Gamma-aminobutyric acid receptor subunit thetaHomo sapiens (human)0.0101

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (83.33)18.2507
2000's1 (16.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Clissold, DB; Ferkany, JW; Pontecorvo, MJ; White, MF1
Tortella, FC; Witkin, JM1
Balster, RL; Bobelis, DJ1
Balster, RL; Cristello, AF; Wiley, JL1
Treiman, DM; Walton, NY1
Balster, RL; Wiley, JL1

Reviews

1 review(s) available for npc 12626 and diazepam

ArticleYear
Rational polytherapy in the treatment of status epilepticus.
    Epilepsy research. Supplement, 1996, Volume: 11

    Topics: Amino Acids; Animals; Anticonvulsants; Brain; Diazepam; Drug Interactions; Drug Synergism; Drug Therapy, Combination; Electroencephalography; Excitatory Amino Acid Antagonists; Humans; Phenytoin; Rats; Receptors, Neurotransmitter; Status Epilepticus

1996

Other Studies

5 other study(ies) available for npc 12626 and diazepam

ArticleYear
N-methyl-D-aspartate antagonists and working memory performance: comparison with the effects of scopolamine, propranolol, diazepam, and phenylisopropyladenosine.
    Behavioral neuroscience, 1991, Volume: 105, Issue:4

    Topics: Amino Acids; Animals; Appetitive Behavior; Brain; Diazepam; Discrimination Learning; Dizocilpine Maleate; Dose-Response Relationship, Drug; Male; Mental Recall; Phencyclidine; Phenylisopropyladenosine; Piperazines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, N-Methyl-D-Aspartate; Receptors, Purinergic; Retention, Psychology; Scopolamine

1991
Modulators of N-methyl-D-aspartate protect against diazepam- or phenobarbital-resistant cocaine convulsions.
    Life sciences, 1991, Volume: 48, Issue:11

    Topics: Amino Acids; Animals; Anticonvulsants; Cocaine; Diazepam; Dizocilpine Maleate; Male; Mice; Phencyclidine; Phenobarbital; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Time Factors

1991
Pharmacological specificity of the discriminative stimulus properties of 2-amino-4,5-(1,2-cyclohexyl)-7-phosphono-heptanoic acid (NPC 12626), a competitive N-methyl-D-aspartate receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2

    Topics: Amino Acids; Animals; Binding, Competitive; Conditioning, Operant; Diazepam; Discrimination Learning; Generalization, Stimulus; Male; Phencyclidine; Pipecolic Acids; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

1993
Effects of site-selective NMDA receptor antagonists in an elevated plus-maze model of anxiety in mice.
    European journal of pharmacology, 1995, Dec-27, Volume: 294, Issue:1

    Topics: Amino Acids; Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Modulators; Male; Mice; Mice, Inbred ICR; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Phencyclidine; Punishment; Quinoxalines; Rats; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate

1995
Effects of modulators of N-methyl-D-aspartate receptor-mediated neurotransmission on diazepam discrimination in rats.
    Life sciences, 2004, May-28, Volume: 75, Issue:2

    Topics: Amino Acids; Animals; Biguanides; Binding Sites; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Agonists; Male; N-Methylaspartate; Pentobarbital; Phencyclidine; Piperazines; Quinolones; Quinoxalines; Rats; Rats, Sprague-Dawley; Riluzole

2004