l 158809 and pd 123319
l 158809 has been researched along with pd 123319 in 12 studies
Compound Research Comparison
Studies (l 158809) | Trials (l 158809) | Recent Studies (post-2010) (l 158809) | Studies (pd 123319) | Trials (pd 123319) | Recent Studies (post-2010) (pd 123319) |
---|---|---|---|---|---|
137 | 0 | 7 | 894 | 6 | 175 |
Protein Interaction Comparison
Protein | Taxonomy | l 158809 (IC50) | pd 123319 (IC50) |
---|---|---|---|
Type-1A angiotensin II receptor | Rattus norvegicus (Norway rat) | 0.21 | |
Type-1B angiotensin II receptor | Rattus norvegicus (Norway rat) | 0.21 | |
Type-2 angiotensin II receptor | Rattus norvegicus (Norway rat) | 0.21 |
Research
Studies (12)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 4 (33.33) | 18.2507 |
2000's | 7 (58.33) | 29.6817 |
2010's | 1 (8.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
---|---|
Bossé, R; Boulay, G; Escher, E; Guillemette, G; Servant, G; Zhou, LM | 1 |
Carretero, OA; Liu, YH; Nass, O; Peterson, E; Sabbah, HN; Sharov, VG; Yang, XP | 1 |
Egashira, K; Shimokawa, H; Tada, H; Takemoto, M; Takeshita, A; Ueno, H; Yamamoto, M | 1 |
Cox, BE; Kaiser, JR; Rosenfeld, CR; Roy, TA | 1 |
Clark, KE; Greenberg, SG; Lambers, DS | 1 |
Li, X; Papp, M; Uhal, BD; Wang, R; Zhuang, J | 1 |
Carretero, OA; Garvin, JL; Ren, Y | 1 |
Cohen, EP; Fish, BL; Moulder, JE | 1 |
Avedanian, L; Bkaily, G; D'Orleans-Juste, P; El-Bizri, N; Gobeil, F; Hazzouri, KM; Jacques, D; Nader, M; Regoli, D; Riopel, J | 1 |
Cohen, EP; Fish, BL; Li, XA; Moulder, JE; Sharma, M | 1 |
Anan, A; Irie, M; Iwata, K; Sakisaka, S; Shakado, S; Sohda, T; Takeyama, Y | 1 |
Chitravanshi, VC; Sapru, HN | 1 |
Other Studies
12 other study(ies) available for l 158809 and pd 123319
Article | Year |
---|---|
Sar1-p-benzoylphenylalanine-angiotensin, a new photoaffinity probe for selective labeling of the type 2 angiotensin receptor.
Topics: Adrenal Cortex; Affinity Labels; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Aorta; Binding, Competitive; Cattle; Cells, Cultured; Female; Humans; Imidazoles; In Vitro Techniques; Myometrium; Pyridines; Rabbits; Receptors, Angiotensin; Tetrazoles; Zona Glomerulosa | 1993 |
Effects of angiotensin-converting enzyme inhibitors and angiotensin II type 1 receptor antagonists in rats with heart failure. Role of kinins and angiotensin II type 2 receptors.
Topics: Angiotensin Receptor Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Bradykinin; Bradykinin Receptor Antagonists; Cardiovascular System; Disease Models, Animal; Drug Interactions; Heart Failure; Imidazoles; Kinins; Male; Models, Cardiovascular; Myocardial Infarction; Myocardium; Pyridines; Ramipril; Rats; Rats, Inbred Lew; Receptor, Angiotensin, Type 1; Tetrazoles | 1997 |
Glibenclamide, a specific inhibitor of ATP-sensitive K+ channels, inhibits coronary vasodilation induced by angiotensin II-receptor antagonists.
Topics: Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Coronary Circulation; Coronary Vessels; Dogs; Enzyme Inhibitors; Glyburide; Hypoglycemic Agents; Imidazoles; NG-Nitroarginine Methyl Ester; Potassium Channel Blockers; Pyridines; Tetrazoles; Vasodilation | 1997 |
Differential development of umbilical and systemic arteries. I. ANG II receptor subtype expression.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Blood Pressure; Cell Membrane; Dose-Response Relationship, Drug; Femoral Artery; Heart Rate; Imidazoles; Muscle, Smooth, Vascular; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Renin; Sheep; Tetrazoles; Umbilical Arteries | 1998 |
Functional role of angiotensin II type 1 and 2 receptors in regulation of uterine blood flow in nonpregnant sheep.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Female; Imidazoles; Injections, Intra-Arterial; Injections, Intravenous; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Regional Blood Flow; Sheep; Tetrazoles; Uterus; Vasoconstriction; Vasoconstrictor Agents | 2000 |
Angiotensin receptor subtype AT(1) mediates alveolar epithelial cell apoptosis in response to ANG II.
Topics: Adenocarcinoma; Angiotensin II; Angiotensin Receptor Antagonists; Antihypertensive Agents; Apoptosis; Cysteine Proteinase Inhibitors; Dose-Response Relationship, Drug; Epithelial Cells; Humans; Imidazoles; Losartan; Lung Neoplasms; Pulmonary Alveoli; Pulmonary Fibrosis; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Respiratory Mucosa; Tetrazoles; Tumor Cells, Cultured; Vasoconstrictor Agents | 2002 |
Vasodilator action of angiotensin-(1-7) on isolated rabbit afferent arterioles.
Topics: Afferent Pathways; Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Arterioles; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Kidney Glomerulus; Male; Norepinephrine; Peptide Fragments; Pyridines; Rabbits; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Tetrazoles; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents | 2002 |
Impact of angiotensin II type 2 receptor blockade on experimental radiation nephropathy.
Topics: Angiotensin II Type 1 Receptor Blockers; Angiotensin II Type 2 Receptor Blockers; Animals; Dose-Response Relationship, Drug; Drug Interactions; Imidazoles; Kidney Diseases; Kidney Function Tests; Male; Pyridines; Radiation Injuries, Experimental; Radiation Protection; Radiation Tolerance; Rats; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Tetrazoles; Treatment Outcome | 2004 |
Angiotensin II induced increase in frequency of cytosolic and nuclear calcium waves of heart cells via activation of AT1 and AT2 receptors.
Topics: Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Angiotensin II Type 2 Receptor Blockers; Animals; Calcium; Calcium Signaling; Cell Nucleus; Chickens; Cytosol; Dose-Response Relationship, Drug; Heart Ventricles; Imidazoles; Indoles; Maleimides; Microscopy, Confocal; Myocytes, Cardiac; Phorbol 12,13-Dibutyrate; Protein Kinase C; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Tetrazoles; Time Factors; Ventricular Function | 2005 |
Role of the angiotensin II type-2 receptor in radiation nephropathy.
Topics: Angiotensin II; Angiotensin II Type 2 Receptor Blockers; Animals; Cell Line; Humans; Imidazoles; Kidney Diseases; Male; Mice; Pyridines; Radiation Injuries, Experimental; Rats; Receptor, Angiotensin, Type 2; Tetrazoles; Time Factors | 2007 |
Angiotensin II type 1 receptor antagonist improves the prognosis in rats displaying liver cirrhosis induced by a choline-deficient diet.
Topics: Angiotensin II; Angiotensin II Type 2 Receptor Blockers; Animals; Antihypertensive Agents; Choline; Disease Models, Animal; Imidazoles; Lipid Peroxidation; Liver Cirrhosis; Male; Pyridines; Rats; Rats, Inbred F344; Tetrazoles; Vasoconstrictor Agents | 2008 |
Cardiovascular responses elicited by a new endogenous angiotensin in the nucleus tractus solitarius of the rat.
Topics: Analysis of Variance; Angiotensin Receptor Antagonists; Angiotensinogen; Angiotensins; Animals; Blood Pressure; Heart Rate; Imidazoles; Male; Microinjections; Naphthyridines; Neurons; Peptide Fragments; Pyridines; Rats; Rats, Wistar; Solitary Nucleus; Splanchnic Nerves; Tetrazoles; Vagotomy | 2011 |