Page last updated: 2024-09-03

indatraline and cep-32496

indatraline has been researched along with cep-32496 in 2 studies

Compound Research Comparison

Studies
(indatraline)
Trials
(indatraline)
Recent Studies (post-2010)
(indatraline)
Studies
(cep-32496)
Trials
(cep-32496)
Recent Studies (post-2010) (cep-32496)
4602418016

Protein Interaction Comparison

ProteinTaxonomyindatraline (IC50)cep-32496 (IC50)
Tyrosine-protein kinase ABL1Homo sapiens (human)0.006
RAF proto-oncogene serine/threonine-protein kinaseHomo sapiens (human)0.146
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)0.0543
Serine/threonine-protein kinase B-rafHomo sapiens (human)0.082
Ephrin type-A receptor 2Homo sapiens (human)0.028
Cytochrome P450 2C19Homo sapiens (human)3.4
Vascular endothelial growth factor receptor 2Homo sapiens (human)0.03
Nuclear receptor coactivator 4Homo sapiens (human)0.0004
Coiled-coil domain-containing protein 6Homo sapiens (human)0.0037

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Kabir, M; Kerns, E; Nguyen, K; Shah, P; Sun, H; Wang, Y; Xu, X; Yu, KR1
Kabir, M; Kerns, E; Neyra, J; Nguyen, K; Nguyễn, ÐT; Shah, P; Siramshetty, VB; Southall, N; Williams, J; Xu, X; Yu, KR1

Other Studies

2 other study(ies) available for indatraline and cep-32496

ArticleYear
Predictive models of aqueous solubility of organic compounds built on A large dataset of high integrity.
    Bioorganic & medicinal chemistry, 2019, 07-15, Volume: 27, Issue:14

    Topics: Drug Discovery; Organic Chemicals; Pharmaceutical Preparations; Solubility

2019
Retrospective assessment of rat liver microsomal stability at NCATS: data and QSAR models.
    Scientific reports, 2020, 11-26, Volume: 10, Issue:1

    Topics: Animals; Computer Simulation; Databases, Factual; Drug Discovery; High-Throughput Screening Assays; Liver; Machine Learning; Male; Microsomes, Liver; National Center for Advancing Translational Sciences (U.S.); Pharmaceutical Preparations; Quantitative Structure-Activity Relationship; Rats; Rats, Sprague-Dawley; Retrospective Studies; United States

2020