Page last updated: 2024-09-03

gbr 13069 and vanoxerine

gbr 13069 has been researched along with vanoxerine in 2 studies

Compound Research Comparison

Studies
(gbr 13069)
Trials
(gbr 13069)
Recent Studies (post-2010)
(gbr 13069)
Studies
(vanoxerine)
Trials
(vanoxerine)
Recent Studies (post-2010) (vanoxerine)
600556593
60028020

Protein Interaction Comparison

ProteinTaxonomygbr 13069 (IC50)vanoxerine (IC50)
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.46
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.0103
Sodium-dependent serotonin transporterHomo sapiens (human)3.84
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.0969
Small conductance calcium-activated potassium channel protein 2Rattus norvegicus (Norway rat)0.073
Small conductance calcium-activated potassium channel protein 3Rattus norvegicus (Norway rat)0.073
Small conductance calcium-activated potassium channel protein 1Rattus norvegicus (Norway rat)0.073
Sodium-dependent dopamine transporter Homo sapiens (human)0.1485
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.022
TransporterRattus norvegicus (Norway rat)0.114
Mu-type opioid receptorHomo sapiens (human)3.53
Kappa-type opioid receptorHomo sapiens (human)2.14

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19901 (50.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Heikkila, RE; Manzino, L1
Grundt, P; Katz, JL; Kopajtic, T; Kulkarni, SS; Newman, AH1

Other Studies

2 other study(ies) available for gbr 13069 and vanoxerine

ArticleYear
Behavioral properties of GBR 12909, GBR 13069 and GBR 13098: specific inhibitors of dopamine uptake.
    European journal of pharmacology, 1984, Aug-17, Volume: 103, Issue:3-4

    Topics: Animals; Behavior, Animal; Biogenic Amines; Cerebral Cortex; Corpus Striatum; Dopamine; Female; Flunarizine; Haloperidol; Humans; Hydroxydopamines; In Vitro Techniques; Male; Mice; Motor Activity; Neurotransmitter Uptake Inhibitors; Oxidopamine; Piperazines; Rats; Rats, Inbred Strains; Stereotyped Behavior

1984
Structure-activity relationships at monoamine transporters for a series of N-substituted 3alpha-(bis[4-fluorophenyl]methoxy)tropanes: comparative molecular field analysis, synthesis, and pharmacological evaluation.
    Journal of medicinal chemistry, 2004, Jun-17, Volume: 47, Issue:13

    Topics: Animals; Brain; Carrier Proteins; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; In Vitro Techniques; Male; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Nerve Tissue Proteins; Norepinephrine Plasma Membrane Transport Proteins; Protein Binding; Quantitative Structure-Activity Relationship; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Serotonin Plasma Membrane Transport Proteins; Symporters; Tropanes

2004
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