Page last updated: 2024-09-04

eglumetad and amphetamine

eglumetad has been researched along with amphetamine in 4 studies

Compound Research Comparison

Studies
(eglumetad)
Trials
(eglumetad)
Recent Studies (post-2010)
(eglumetad)
Studies
(amphetamine)
Trials
(amphetamine)
Recent Studies (post-2010) (amphetamine)
19054813,0713291,977

Protein Interaction Comparison

ProteinTaxonomyeglumetad (IC50)amphetamine (IC50)
Phenylethanolamine N-methyltransferaseBos taurus (cattle)0.96
Cytochrome P450 2A6Homo sapiens (human)3.5
Cytochrome P450 2A5Mus musculus (house mouse)2.85
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.96
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.96

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's3 (75.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Guo, N; Huang, Y; Hwang, DR; Kegeles, LS; Laruelle, M; Narendran, R; van Berckel, BN; Van Heertum, R; Waterhouse, R1
Moghaddam, B; Pehrson, AL1
Gibula-Bruzda, E; Koltunowska, D; Kotlinska, JH1
Hewes, N; Lodge, D; McCarthy, AP; Robinson, ESJ; Shanks, E; Wafford, KA; Wood, CM1

Other Studies

4 other study(ies) available for eglumetad and amphetamine

ArticleYear
Modulation of amphetamine-induced dopamine release by group II metabotropic glutamate receptor agonist LY354740 in non-human primates studied with positron emission tomography.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2006, Volume: 31, Issue:5

    Topics: Amphetamine; Animals; Brain; Bridged Bicyclo Compounds; Dopamine; Dopamine Agents; Dopamine Antagonists; Excitatory Amino Acid Agonists; Female; Male; Papio anubis; Positron-Emission Tomography; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Schizophrenia

2006
Impact of metabotropic glutamate 2/3 receptor stimulation on activated dopamine release and locomotion.
    Psychopharmacology, 2010, Volume: 211, Issue:4

    Topics: Amphetamine; Animals; Bridged Bicyclo Compounds; Dopamine; Electric Stimulation; Excitatory Amino Acid Agonists; Extracellular Space; Levodopa; Locomotion; Male; Microdialysis; Neurons; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate

2010
The influence of ionotropic and metabotropic glutamate receptor ligands on anxiety-like effect of amphetamine withdrawal in rats.
    Progress in neuro-psychopharmacology & biological psychiatry, 2013, Aug-01, Volume: 45

    Topics: Acamprosate; Amphetamine; Animals; Anxiety; Bridged Bicyclo Compounds; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Ligands; Male; Memantine; Pyridines; Rats; Receptors, Ionotropic Glutamate; Receptors, Metabotropic Glutamate; Substance Withdrawal Syndrome; Taurine; Thiazoles

2013
Investigating the role of mGluR2 versus mGluR3 in antipsychotic-like effects, sleep-wake architecture and network oscillatory activity using novel Han Wistar rats lacking mGluR2 expression.
    Neuropharmacology, 2018, 09-15, Volume: 140

    Topics: Amino Acids; Amphetamine; Animals; Antipsychotic Agents; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cyclohexanes; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Gamma Rhythm; Locomotion; Male; Motor Activity; Mutation; Phencyclidine; Rats; Receptors, Metabotropic Glutamate; Sleep; Theta Rhythm; Wakefulness

2018