Page last updated: 2024-09-03

cgp 361a and reserpine

cgp 361a has been researched along with reserpine in 3 studies

Compound Research Comparison

Studies
(cgp 361a)
Trials
(cgp 361a)
Recent Studies (post-2010)
(cgp 361a)
Studies
(reserpine)
Trials
(reserpine)
Recent Studies (post-2010) (reserpine)
213315,546223436

Protein Interaction Comparison

ProteinTaxonomycgp 361a (IC50)reserpine (IC50)
Bile salt export pumpHomo sapiens (human)8.7875
ATP-dependent translocase ABCB1Homo sapiens (human)3.2092
Quinolone resistance protein NorAStaphylococcus aureus8.5429
Mu-type opioid receptorHomo sapiens (human)4.152
Chromaffin granule amine transporterHomo sapiens (human)0.05
Synaptic vesicular amine transporterRattus norvegicus (Norway rat)0.0034
Synaptic vesicular amine transporterHomo sapiens (human)0.0147

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19901 (33.33)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baumann, PA; Bischoff, S; Neale, RF; Sills, MA; Waldmeier, PC; Williams, M1
Atack, J; Chadha, A; Duty, S; Sur, C1
Ahlenius, S; Kaur, P1

Other Studies

3 other study(ies) available for cgp 361a and reserpine

ArticleYear
Interactions of isamoltane (CGP 361A), an anxiolytic phenoxypropanolamine derivative, with 5-HT1 receptor subtypes in the rat brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 337, Issue:6

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Anti-Anxiety Agents; Brain; Cerebral Cortex; Corpus Striatum; Electric Stimulation; Hippocampus; In Vitro Techniques; Iodocyanopindolol; Male; Pindolol; Propanolamines; Rats; Receptors, Serotonin; Reserpine; Serotonin; Stereoisomerism; Tetrahydronaphthalenes

1988
The 5HT(1B) receptor agonist, CP-93129, inhibits [(3)H]-GABA release from rat globus pallidus slices and reverses akinesia following intrapallidal injection in the reserpine-treated rat.
    British journal of pharmacology, 2000, Volume: 130, Issue:8

    Topics: Animals; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Globus Pallidus; In Vitro Techniques; Male; Movement Disorders; Propanolamines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reserpine; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium

2000
Non-serotonergic potentiation by (-)-pindolol of DOI-induced forward locomotion in rats: possible involvement of beta-adrenoceptors?.
    Journal of neural transmission (Vienna, Austria : 1996), 2000, Volume: 107, Issue:8-9

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Animals; Betaxolol; Biogenic Monoamines; Dihydroxyphenylalanine; Drug Synergism; Indophenol; Male; Motor Activity; Pindolol; Piperazines; Piperidines; Propanolamines; Prosencephalon; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Adrenergic, beta; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reserpine; Serotonin Antagonists; Serotonin Receptor Agonists

2000