anatoxin a has been researched along with cytisine in 5 studies
Studies (anatoxin a) | Trials (anatoxin a) | Recent Studies (post-2010) (anatoxin a) | Studies (cytisine) | Trials (cytisine) | Recent Studies (post-2010) (cytisine) |
---|---|---|---|---|---|
522 | 0 | 126 | 519 | 19 | 178 |
6 | 0 | 1 | 519 | 19 | 178 |
Protein | Taxonomy | anatoxin a (IC50) | cytisine (IC50) |
---|---|---|---|
Neuronal acetylcholine receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | 0.0692 | |
Neuronal acetylcholine receptor subunit beta-2 | Rattus norvegicus (Norway rat) | 0.0692 | |
Neuronal acetylcholine receptor subunit beta-2 | Homo sapiens (human) | 0.05 | |
Neuronal acetylcholine receptor subunit alpha-4 | Homo sapiens (human) | 0.05 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (60.00) | 18.2507 |
2000's | 1 (20.00) | 29.6817 |
2010's | 1 (20.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Dart, MJ; Holladay, MW; Lynch, JK | 1 |
Gohlke, H; Gündisch, D; Schwarz, S; Seitz, G; Tilotta, MC; Weber, A; Wegge, T | 1 |
Amar, M; Johnson, C; Lunt, GG; Thomas, P; Wonnacott, S | 1 |
Clarke, PB; Reuben, M | 1 |
Fasoli, F; Gotti, C; Novelli, F; Sparatore, F; Tasso, B | 1 |
1 review(s) available for anatoxin a and cytisine
Article | Year |
---|---|
Neuronal nicotinic acetylcholine receptors as targets for drug discovery.
Topics: Acetylcholine; Animals; Binding Sites; Dopamine; Drug Design; Humans; Molecular Structure; Nervous System; Neurons; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Receptors, Nicotinic; Structure-Activity Relationship | 1997 |
4 other study(ies) available for anatoxin a and cytisine
Article | Year |
---|---|
3D QSAR analyses-guided rational design of novel ligands for the (alpha4)2(beta2)3 nicotinic acetylcholine receptor.
Topics: Alkaloids; Animals; Azocines; Bacterial Toxins; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cyanobacteria Toxins; Drug Design; In Vitro Techniques; Ligands; Marine Toxins; Microcystins; Models, Molecular; Prosencephalon; Protein Subunits; Pyridines; Quantitative Structure-Activity Relationship; Quinolizines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Stereoisomerism; Tropanes | 2003 |
Agonist pharmacology of the neuronal alpha 7 nicotinic receptor expressed in Xenopus oocytes.
Topics: Acetylcholine; Alkaloids; Animals; Azocines; Bacterial Toxins; Cyanobacteria Toxins; Dimethylphenylpiperazinium Iodide; DNA; Marine Toxins; Membrane Potentials; Microcystins; Neurons; Nicotine; Oocytes; Piperazines; Quaternary Ammonium Compounds; Quinolizines; Receptors, Nicotinic; Tropanes; Xenopus | 1993 |
Release of [3H]-noradrenaline from rat hippocampal synaptosomes by nicotine: mediation by different nicotinic receptor subtypes from striatal [3H]-dopamine release.
Topics: Acetylcholine; Alkaloids; Animals; Azocines; Bacterial Toxins; Citalopram; Corpus Striatum; Cyanobacteria Toxins; Hippocampus; In Vitro Techniques; Male; Marine Toxins; Microcystins; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Norepinephrine; Potassium; Quinolizines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Serotonin Antagonists; Synaptosomes; Tetrodotoxin; Tritium; Tropanes | 1996 |
(+)-Laburnamine, a natural selective ligand and partial agonist for the α4β2 nicotinic receptor subtype.
Topics: Alkaloids; Animals; Binding, Competitive; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Humans; Italy; Ligands; Neostriatum; Nicotine; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Seeds; Stereoisomerism | 2013 |