Page last updated: 2024-09-02

anatoxin a and cytisine

anatoxin a has been researched along with cytisine in 5 studies

Compound Research Comparison

Studies
(anatoxin a)
Trials
(anatoxin a)
Recent Studies (post-2010)
(anatoxin a)
Studies
(cytisine)
Trials
(cytisine)
Recent Studies (post-2010) (cytisine)
522012651919178
60151919178

Protein Interaction Comparison

ProteinTaxonomyanatoxin a (IC50)cytisine (IC50)
Neuronal acetylcholine receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0692
Neuronal acetylcholine receptor subunit beta-2Rattus norvegicus (Norway rat)0.0692
Neuronal acetylcholine receptor subunit beta-2Homo sapiens (human)0.05
Neuronal acetylcholine receptor subunit alpha-4Homo sapiens (human)0.05

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (60.00)18.2507
2000's1 (20.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dart, MJ; Holladay, MW; Lynch, JK1
Gohlke, H; Gündisch, D; Schwarz, S; Seitz, G; Tilotta, MC; Weber, A; Wegge, T1
Amar, M; Johnson, C; Lunt, GG; Thomas, P; Wonnacott, S1
Clarke, PB; Reuben, M1
Fasoli, F; Gotti, C; Novelli, F; Sparatore, F; Tasso, B1

Reviews

1 review(s) available for anatoxin a and cytisine

ArticleYear
Neuronal nicotinic acetylcholine receptors as targets for drug discovery.
    Journal of medicinal chemistry, 1997, Dec-19, Volume: 40, Issue:26

    Topics: Acetylcholine; Animals; Binding Sites; Dopamine; Drug Design; Humans; Molecular Structure; Nervous System; Neurons; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Receptors, Nicotinic; Structure-Activity Relationship

1997

Other Studies

4 other study(ies) available for anatoxin a and cytisine

ArticleYear
3D QSAR analyses-guided rational design of novel ligands for the (alpha4)2(beta2)3 nicotinic acetylcholine receptor.
    Journal of medicinal chemistry, 2003, May-22, Volume: 46, Issue:11

    Topics: Alkaloids; Animals; Azocines; Bacterial Toxins; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cyanobacteria Toxins; Drug Design; In Vitro Techniques; Ligands; Marine Toxins; Microcystins; Models, Molecular; Prosencephalon; Protein Subunits; Pyridines; Quantitative Structure-Activity Relationship; Quinolizines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Stereoisomerism; Tropanes

2003
Agonist pharmacology of the neuronal alpha 7 nicotinic receptor expressed in Xenopus oocytes.
    FEBS letters, 1993, Aug-02, Volume: 327, Issue:3

    Topics: Acetylcholine; Alkaloids; Animals; Azocines; Bacterial Toxins; Cyanobacteria Toxins; Dimethylphenylpiperazinium Iodide; DNA; Marine Toxins; Membrane Potentials; Microcystins; Neurons; Nicotine; Oocytes; Piperazines; Quaternary Ammonium Compounds; Quinolizines; Receptors, Nicotinic; Tropanes; Xenopus

1993
Release of [3H]-noradrenaline from rat hippocampal synaptosomes by nicotine: mediation by different nicotinic receptor subtypes from striatal [3H]-dopamine release.
    British journal of pharmacology, 1996, Volume: 117, Issue:4

    Topics: Acetylcholine; Alkaloids; Animals; Azocines; Bacterial Toxins; Citalopram; Corpus Striatum; Cyanobacteria Toxins; Hippocampus; In Vitro Techniques; Male; Marine Toxins; Microcystins; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Norepinephrine; Potassium; Quinolizines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Serotonin Antagonists; Synaptosomes; Tetrodotoxin; Tritium; Tropanes

1996
(+)-Laburnamine, a natural selective ligand and partial agonist for the α4β2 nicotinic receptor subtype.
    Journal of natural products, 2013, Apr-26, Volume: 76, Issue:4

    Topics: Alkaloids; Animals; Binding, Competitive; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Humans; Italy; Ligands; Neostriatum; Nicotine; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Seeds; Stereoisomerism

2013