Page last updated: 2024-09-05

a 69024 and spiperone

a 69024 has been researched along with spiperone in 3 studies

Compound Research Comparison

Studies
(a 69024)
Trials
(a 69024)
Recent Studies (post-2010)
(a 69024)
Studies
(spiperone)
Trials
(spiperone)
Recent Studies (post-2010) (spiperone)
13002,9441385

Protein Interaction Comparison

ProteinTaxonomya 69024 (IC50)spiperone (IC50)
Bile salt export pumpHomo sapiens (human)10
D(2) dopamine receptorHomo sapiens (human)0.0008
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.097
D(4) dopamine receptorHomo sapiens (human)0.0005
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.097
Histamine H1 receptorCavia porcellus (domestic guinea pig)0.097
D(3) dopamine receptorHomo sapiens (human)0.0635
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.097
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0001
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.955

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's2 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bals-Kubik, R; Herz, A; Huber, A; Shippenberg, TS1
Dikic, B; Kassiou, M; Katsifis, A; Mardon, K; Mattner, F1
DeJesus, OT; Gatley, SJ; Gifford, AN; Huemmer, CL; Rice, OV; Rogoz, R; Shen, J; Volkow, ND1

Other Studies

3 other study(ies) available for a 69024 and spiperone

ArticleYear
Neuroanatomical substrates mediating the aversive effects of D-1 dopamine receptor antagonists.
    Psychopharmacology, 1991, Volume: 103, Issue:2

    Topics: Animals; Benzazepines; Brain; Dopamine Antagonists; Injections, Intraventricular; Limbic System; Male; Microinjections; Papaverine; Rats; Rats, Inbred Strains; Receptors, Dopamine D1; Spiperone; Stereotaxic Techniques; Sulpiride; Tetrahydroisoquinolines

1991
Pharmacological evaluation of (+)-2- [123I]A-69024: a radioligand for in vivo studies of dopamine D1 receptors.
    Life sciences, 2001, Jun-29, Volume: 69, Issue:6

    Topics: Animals; Benzazepines; Brain; Cerebellum; Clozapine; Corpus Striatum; Dopamine Antagonists; Haloperidol; Injections, Intravenous; Iodine Radioisotopes; Ketanserin; Ligands; Male; Papaverine; Rats; Rats, Wistar; Receptors, Dopamine D1; Spiperone; Stereoisomerism; Tetrahydroisoquinolines; Tetrahydronaphthalenes; Tissue Distribution; Tomography, Emission-Computed, Single-Photon

2001
Effects of endogenous neurotransmitters on the in vivo binding of dopamine and 5-HT radiotracers in mice.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2001, Volume: 25, Issue:5

    Topics: Animals; Binding, Competitive; Dopamine; Dopamine Agonists; Dopamine Antagonists; Male; Mice; Neurotransmitter Agents; Papaverine; Piperazines; Pyridines; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D1; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Spiperone; Tetrahydroisoquinolines

2001