Page last updated: 2024-08-05 15:49:09

SERCA activator

Any compound that activates Sarcoplasmic/Endoplasmic Reticulum Calcium-ATPase (EC 7.2.2.10).

ChEBI ID: 150006

Members (1)

MemberDefinitionClass
CDN1163A secondary carboxamide resulting from the formal condensation of the carboxy group of 4-isopropoxybenzoic acid with the primary amino group of 2-methylquinolin-8-amine. An allosteric activator of sarco/endoplasmic reticulum Ca(2+)-ATPase (SERCA).CDN1163

Research

Studies (17)

TimeframeStudies, Drugs with This Role(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's8 (47.06)24.3611
2020's9 (52.94)2.80

Study Types

Publication TypeStudies, Drugs with this Role (%)All Drugs (%)
Trials0 (0.00%)5.53%
Reviews0 (0.00%)6.00%
Case Studies0 (0.00%)4.05%
Observational0 (0.00%)0.25%
Other17 (100.00%)84.16%

Protein Targets (4)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
Chain A, Ferritin light chainEquus caballus (horse)Potency0.794311
Single-stranded DNA cytosine deaminaseHomo sapiens (human)Potency39.810711
TAR DNA-binding protein 43Homo sapiens (human)Potency11.220211
TDP1 proteinHomo sapiens (human)Potency23.724622