Proteins > Gamma-aminobutyric acid type B receptor subunit 1
Page last updated: 2024-08-07 13:50:19
Gamma-aminobutyric acid type B receptor subunit 1
A gamma-aminobutyric acid type B receptor subunit 1 that is encoded in the genome of rat. [OMA:Q9Z0U4, PRO:DNx]
Synonyms
GABA-B receptor 1;
GABA-B-R1;
GABA-BR1;
GABABR1;
Gb1
Research
Bioassay Publications (7)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 1 (14.29) | 18.7374 |
| 1990's | 6 (85.71) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (13)
Drugs with Inhibition Measurements
Partial GABAA receptor agonists. Synthesis and in vitro pharmacology of a series of nonannulated analogs of 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
3-Thienyl- and 3-furylaminobutyric acids. Synthesis and binding GABAB receptor studies.Journal of medicinal chemistry, , Volume: 34, Issue:8, 1991
Synthesis and pharmacological evaluation of gamma-aminobutyric acid analogues. New ligand for GABAB sites.Journal of medicinal chemistry, , Volume: 30, Issue:4, 1987
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Synthesis and biochemical evaluation of baclofen analogues locked in the baclofen solid-state conformation.Journal of medicinal chemistry, , Volume: 34, Issue:4, 1991
3-Thienyl- and 3-furylaminobutyric acids. Synthesis and binding GABAB receptor studies.Journal of medicinal chemistry, , Volume: 34, Issue:8, 1991
Synthesis and pharmacological evaluation of gamma-aminobutyric acid analogues. New ligand for GABAB sites.Journal of medicinal chemistry, , Volume: 30, Issue:4, 1987
Phosphinic acid analogues of GABA. 2. Selective, orally active GABAB antagonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Synthesis and pharmacology of the baclofen homologues 5-amino-4-(4-chlorophenyl)pentanoic acid and the R- and S-enantiomers of 5-amino-3-(4-chlorophenyl)pentanoic acid.Journal of medicinal chemistry, , Jun-03, Volume: 42, Issue:11, 1999
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Phosphinic acid analogues of GABA. 2. Selective, orally active GABAB antagonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995