Page last updated: 2024-08-07 17:11:28

Beta-2 adrenergic receptor

A beta-2 adrenergic receptor that is encoded in the genome of cow. [OMA:Q28044, PRO:DNx]

Synonyms

Beta-2 adrenoreceptor;
Beta-2 adrenoceptor

Research

Bioassay Publications (6)

TimeframeStudies on this Protein(%)All Drugs %
pre-19902 (33.33)18.7374
1990's4 (66.67)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (19)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
isoproterenolBos taurus (cattle)Ki0.110022
dichloroisoproterenolBos taurus (cattle)Ki0.140011
panadiplonBos taurus (cattle)Ki0.001611

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
albuterolBos taurus (cattle)Kd0.520011
betaxololBos taurus (cattle)Kd186.210011
clenbuterolBos taurus (cattle)Kd0.036011
isoproterenolBos taurus (cattle)Kd0.330011
metaproterenolBos taurus (cattle)Kd9.120011
practololBos taurus (cattle)Kd20.417011
pronethalolBos taurus (cattle)Kd0.160011
sotalolBos taurus (cattle)Kd0.580011
terbutalineBos taurus (cattle)Kd3.980011
tulobuterolBos taurus (cattle)Kd0.130011
nifenalolBos taurus (cattle)Kd1.320011
toliprololBos taurus (cattle)Kd0.043611
deterenolBos taurus (cattle)Kd4.270011
colterolBos taurus (cattle)Kd0.600011
prenalterolBos taurus (cattle)Kd1.072011
dihydroalprenololBos taurus (cattle)Kd0.000611
propranolol hydrochlorideBos taurus (cattle)Kd0.000911

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
albuterolBos taurus (cattle)Concentration30.000011
albuterolBos taurus (cattle)KD app0.570011
clenbuterolBos taurus (cattle)Concentration1.000011
clenbuterolBos taurus (cattle)KD app0.037011
terbutalineBos taurus (cattle)Concentration1,000,000.000011
terbutalineBos taurus (cattle)KD app4.480011
tulobuterolBos taurus (cattle)Concentration10.000011
tulobuterolBos taurus (cattle)KD app0.130011
colterolBos taurus (cattle)Concentration3,000,000.000011
colterolBos taurus (cattle)KD app0.670011