Page last updated: 2024-08-07 17:11:28
Beta-2 adrenergic receptor
A beta-2 adrenergic receptor that is encoded in the genome of cow. [OMA:Q28044, PRO:DNx]
Synonyms
Beta-2 adrenoreceptor;
Beta-2 adrenoceptor
Research
Bioassay Publications (6)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 2 (33.33) | 18.7374 |
1990's | 4 (66.67) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (19)
Drugs with Inhibition Measurements
Drugs with Activation Measurements
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
albuterol | Bos taurus (cattle) | Concentration | 30.0000 | 1 | 1 |
albuterol | Bos taurus (cattle) | KD app | 0.5700 | 1 | 1 |
clenbuterol | Bos taurus (cattle) | Concentration | 1.0000 | 1 | 1 |
clenbuterol | Bos taurus (cattle) | KD app | 0.0370 | 1 | 1 |
terbutaline | Bos taurus (cattle) | Concentration | 1,000,000.0000 | 1 | 1 |
terbutaline | Bos taurus (cattle) | KD app | 4.4800 | 1 | 1 |
tulobuterol | Bos taurus (cattle) | Concentration | 10.0000 | 1 | 1 |
tulobuterol | Bos taurus (cattle) | KD app | 0.1300 | 1 | 1 |
colterol | Bos taurus (cattle) | Concentration | 3,000,000.0000 | 1 | 1 |
colterol | Bos taurus (cattle) | KD app | 0.6700 | 1 | 1 |
Conformationally restrained analogs of sympathomimetic catecholamines. Synthesis, conformational analysis, and adrenergic activity of isochroman derivatives.Journal of medicinal chemistry, , Oct-15, Volume: 36, Issue:21, 1993
Conformational effects on the activity of drugs. 13. A revision of previously proposed models for the activation of alpha- and beta-adrenergic receptors.Journal of medicinal chemistry, , Mar-20, Volume: 35, Issue:6, 1992
Quantitative evaluation of the beta 2-adrenoceptor affinity of phenoxypropanolamines and phenylethanolamines.Journal of medicinal chemistry, , Volume: 28, Issue:9, 1985