Page last updated: 2024-08-07 16:58:33
Thyrotropin-releasing hormone receptor
A thyrotropin-releasing hormone receptor type 1 that is encoded in the genome of rat. [OMA:Q01717, PRO:DNx]
Synonyms
TRH-R;
Thyroliberin receptor
Research
Bioassay Publications (3)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 1 (33.33) | 18.2507 |
| 2000's | 2 (66.67) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (3)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| ondansetron | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| thyrotropin-releasing hormone | Rattus norvegicus (Norway rat) | Ki | 0.0311 | 2 | 2 |
| cilansetron | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| thyrotropin-releasing hormone | Rattus norvegicus (Norway rat) | EC50 | 0.0030 | 1 | 1 |