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Mycocyclosin synthase

A protein that is a translation product of the cyp121 gene in Mycobacterium tuberculosis H37Rv. [PRO:DNx, UniProtKB:P9WPP7]

Synonyms

EC 1.14.19.70;
Cytochrome P450 121;
Cytochrome P450 MT2

Research

Bioassay Publications (2)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Compounds (4)

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
clotrimazoleMycobacterium tuberculosis H37RvKd0.073011
econazoleMycobacterium tuberculosis H37RvKd0.073011
fluconazoleMycobacterium tuberculosis H37RvKd6.000011
miconazoleMycobacterium tuberculosis H37RvKd0.073011
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