Page last updated: 2024-08-07 15:57:50
Beta-lactamase OXA-1
A protein that is a translation product of any of the plasmid-encoded copies of the bla gene in Escherichia coli. [PRO:DAN, UniProtKB:P13661]
Synonyms
EC 3.5.2.6;
Penicillinase
Research
Bioassay Publications (4)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 1 (25.00) | 18.7374 |
1990's | 1 (25.00) | 18.2507 |
2000's | 2 (50.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (4)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
tazobactam | Escherichia coli | IC50 | 4.8000 | 1 | 1 |
sulbactam | Escherichia coli | IC50 | 22.0000 | 1 | 1 |
clavulanic acid | Escherichia coli | IC50 | 3.2000 | 1 | 1 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
cephalothin | Escherichia coli | Km | 10.0000 | 1 | 1 |
tazobactam | Escherichia coli | Kinact | 380.0000 | 1 | 1 |