Page last updated: 2024-08-07 15:44:56

Neprilysin

A protein that is a translation product of the MME gene in rabbit. [PRO:DNx, UniProtKB:P08049]

Synonyms

EC 3.4.24.11;
Atriopeptidase;
Enkephalinase;
Neutral endopeptidase 24.11;
NEP;
Neutral endopeptidase;
Skin fibroblast elastase;
SFE

Research

Bioassay Publications (8)

TimeframeStudies on this Protein(%)All Drugs %
pre-19904 (50.00)18.7374
1990's3 (37.50)18.2507
2000's1 (12.50)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (9)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
thiorphanOryctolagus cuniculus (rabbit)IC500.008544
thiorphanOryctolagus cuniculus (rabbit)Ki2.527024
captoprilOryctolagus cuniculus (rabbit)Ki3.000524
kelatorphanOryctolagus cuniculus (rabbit)IC500.003633
(3-(n-hydroxy)carboxamido-2-benzylpropanoyl)glycineOryctolagus cuniculus (rabbit)IC500.001422
actinoninOryctolagus cuniculus (rabbit)IC508.200011
phosphoramidonOryctolagus cuniculus (rabbit)IC500.002833
thiorphanOryctolagus cuniculus (rabbit)IC500.001911
thiorphanOryctolagus cuniculus (rabbit)Ki0.001911
sch 32615Oryctolagus cuniculus (rabbit)IC500.020011
cgs 35066Oryctolagus cuniculus (rabbit)IC502.300011